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1.
Discovery of MDV6058 (PF-06952229), a selective and potent TGFßR1 inhibitor: Design, synthesis and optimization.
Bioorg Med Chem Lett
; 75: 128979, 2022 11 01.
Article
in English
| MEDLINE | ID: mdl-36089110
2.
Discovery of Pyrazolopyrimidine Derivatives as Novel Dual Inhibitors of BTK and PI3Kδ.
ACS Med Chem Lett
; 7(12): 1161-1166, 2016 Dec 08.
Article
in English
| MEDLINE | ID: mdl-27994757
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