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1.
Unexpected Single-Ligand Occupancy and Negative Cooperativity in the SARS-CoV-2 Main Protease.
J Chem Inf Model
; 64(3): 892-904, 2024 Feb 12.
Article
in English
| MEDLINE | ID: mdl-38051605
2.
Identification of Novel GSK-3ß Hits Using Competitive Biophysical Assays.
Int J Mol Sci
; 23(7)2022 Mar 31.
Article
in English
| MEDLINE | ID: mdl-35409221
3.
Structural and Biochemical Analysis of the Dual Inhibition of MG-132 against SARS-CoV-2 Main Protease (Mpro/3CLpro) and Human Cathepsin-L.
Int J Mol Sci
; 22(21)2021 Oct 29.
Article
in English
| MEDLINE | ID: mdl-34769210
4.
Known Drugs Identified by Structure-Based Virtual Screening Are Able to Bind Sigma-1 Receptor and Increase Growth of Huntington Disease Patient-Derived Cells.
Int J Mol Sci
; 22(3)2021 Jan 28.
Article
in English
| MEDLINE | ID: mdl-33525510
5.
Emerging SARS-CoV-2 mutation hot spots include a novel RNA-dependent-RNA polymerase variant.
J Transl Med
; 18(1): 179, 2020 04 22.
Article
in English
| MEDLINE | ID: mdl-32321524
6.
Comparative analysis of fusion tags used to functionalize recombinant antibodies.
Protein Expr Purif
; 166: 105505, 2020 02.
Article
in English
| MEDLINE | ID: mdl-31563543
7.
Insight into GEBR-32a: Chiral Resolution, Absolute Configuration and Enantiopreference in PDE4D Inhibition.
Molecules
; 25(4)2020 Feb 19.
Article
in English
| MEDLINE | ID: mdl-32093112
8.
Combination of SAXS and Protein Painting Discloses the Three-Dimensional Organization of the Bacterial Cysteine Synthase Complex, a Potential Target for Enhancers of Antibiotic Action.
Int J Mol Sci
; 20(20)2019 Oct 21.
Article
in English
| MEDLINE | ID: mdl-31640223
9.
Molecular Bases of PDE4D Inhibition by Memory-Enhancing GEBR Library Compounds.
Biochemistry
; 57(19): 2876-2888, 2018 05 15.
Article
in English
| MEDLINE | ID: mdl-29652483
10.
Baculovirus-driven protein expression in insect cells: A benchmarking study.
J Struct Biol
; 203(2): 71-80, 2018 08.
Article
in English
| MEDLINE | ID: mdl-29545204
11.
Topoisomerase IIß mediates the resistance of glioblastoma stem cells to replication stress-inducing drugs.
Cancer Cell Int
; 16: 58, 2016.
Article
in English
| MEDLINE | ID: mdl-27462186
12.
L-serine biosynthesis in the human central nervous system: Structure and function of phosphoserine aminotransferase.
Protein Sci
; 32(4): e4609, 2023 04.
Article
in English
| MEDLINE | ID: mdl-36851825
13.
Identification of additional mechanistically important residues in the multidrug transporter styMdtM of Salmonella Typhi.
J Biomol Struct Dyn
; : 1-10, 2023 Oct 03.
Article
in English
| MEDLINE | ID: mdl-37787617
14.
Broad-spectrum coronavirus 3C-like protease peptidomimetic inhibitors effectively block SARS-CoV-2 replication in cells: Design, synthesis, biological evaluation, and X-ray structure determination.
Eur J Med Chem
; 253: 115311, 2023 May 05.
Article
in English
| MEDLINE | ID: mdl-37043904
15.
Molecular architecture of the glycogen- committed PP1/PTG holoenzyme.
Nat Commun
; 13(1): 6199, 2022 10 19.
Article
in English
| MEDLINE | ID: mdl-36261419
16.
Easy access to α-ketoamides as SARS-CoV-2 and MERS Mpro inhibitors via the PADAM oxidation route.
Eur J Med Chem
; 244: 114853, 2022 Dec 15.
Article
in English
| MEDLINE | ID: mdl-36332546
17.
ARN25068, a versatile starting point towards triple GSK-3ß/FYN/DYRK1A inhibitors to tackle tau-related neurological disorders.
Eur J Med Chem
; 229: 114054, 2022 Feb 05.
Article
in English
| MEDLINE | ID: mdl-34959172
18.
Design, synthesis, biological evaluation and structural characterization of novel GEBR library PDE4D inhibitors.
Eur J Med Chem
; 223: 113638, 2021 Nov 05.
Article
in English
| MEDLINE | ID: mdl-34171658
19.
Binding of tyrosine kinase inhibitor to epidermal growth factor receptor: surface-enhanced infrared absorption microscopy reveals subtle protein secondary structure variations.
Nanoscale
; 13(16): 7667-7677, 2021 Apr 30.
Article
in English
| MEDLINE | ID: mdl-33928964
20.
An anti-HER2 nanobody binds to its antigen HER2 via two independent paratopes.
Int J Biol Macromol
; 182: 502-511, 2021 Jul 01.
Article
in English
| MEDLINE | ID: mdl-33848543