Detalles de la búsqueda
1.
Value of 68Ga-labeled bombesin antagonist (RM2) in the detection of primary prostate cancer comparing with [18F]fluoromethylcholine PET-CT and multiparametric MRI-a phase I/II study.
Eur Radiol
; 33(1): 472-482, 2023 Jan.
Artículo
en Inglés
| MEDLINE | ID: mdl-35864350
2.
18F-FSPG PET/CT Imaging of System xC- Transporter Activity in Patients with Primary and Metastatic Brain Tumors.
Radiology
; 303(3): 620-631, 2022 06.
Artículo
en Inglés
| MEDLINE | ID: mdl-35191738
3.
Structure-activity relationship around PI-2620 highlights the importance of the nitrogen atom position in the tricyclic core.
Bioorg Med Chem
; 52: 116528, 2021 12 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-34839158
4.
Discovery and preclinical characterization of [18F]PI-2620, a next-generation tau PET tracer for the assessment of tau pathology in Alzheimer's disease and other tauopathies.
Eur J Nucl Med Mol Imaging
; 46(10): 2178-2189, 2019 Sep.
Artículo
en Inglés
| MEDLINE | ID: mdl-31264169
5.
Radiotracer stereochemistry affects substrate affinity and kinetics for improved imaging of system xC- in tumors.
Theranostics
; 12(4): 1921-1936, 2022.
Artículo
en Inglés
| MEDLINE | ID: mdl-35198080
6.
68Ga-Radiolabeling and Pharmacological Characterization of a Kit-Based Formulation of the Gastrin-Releasing Peptide Receptor (GRP-R) Antagonist RM2 for Convenient Preparation of [68Ga]Ga-RM2.
Pharmaceutics
; 13(8)2021 Jul 28.
Artículo
en Inglés
| MEDLINE | ID: mdl-34452121
7.
GMP-Compliant Radiosynthesis of [18F]GP1, a Novel PET Tracer for the Detection of Thrombi.
Pharmaceuticals (Basel)
; 14(8)2021 Jul 28.
Artículo
en Inglés
| MEDLINE | ID: mdl-34451836
8.
PI-2620 Lead Optimization Highlights the Importance of Off-Target Assays to Develop a PET Tracer for the Detection of Pathological Aggregated Tau in Alzheimer's Disease and Other Tauopathies.
J Med Chem
; 64(17): 12808-12830, 2021 09 09.
Artículo
en Inglés
| MEDLINE | ID: mdl-34455780
9.
On the consensus nomenclature rules for radiopharmaceutical chemistry - Reconsideration of radiochemical conversion.
Nucl Med Biol
; 93: 19-21, 2021 02.
Artículo
en Inglés
| MEDLINE | ID: mdl-33232876
10.
Initial evaluation of (4S)-4-(3-[18F]fluoropropyl)-L-glutamate (FSPG) PET/CT imaging in patients with head and neck cancer, colorectal cancer, or non-Hodgkin lymphoma.
EJNMMI Res
; 10(1): 100, 2020 Aug 28.
Artículo
en Inglés
| MEDLINE | ID: mdl-32857284
11.
Discovery of 2-(4-(2-fluoroethoxy)piperidin-1-yl)-9-methyl-9H-pyrrolo[2,3-b:4,5-c']dipyridine ([18F]PI-2014) as PET tracer for the detection of pathological aggregated tau in Alzheimer's disease and other tauopathies.
Eur J Med Chem
; 204: 112615, 2020 Oct 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-32771872
12.
Clinical Evaluation of (4S)-4-(3-[18F]Fluoropropyl)-L-glutamate (18F-FSPG) for PET/CT Imaging in Patients with Newly Diagnosed and Recurrent Prostate Cancer.
Clin Cancer Res
; 26(20): 5380-5387, 2020 10 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-32694158
13.
Tau PET imaging with 18F-PI-2620 in Patients with Alzheimer Disease and Healthy Controls: A First-in-Humans Study.
J Nucl Med
; 61(6): 911-919, 2020 06.
Artículo
en Inglés
| MEDLINE | ID: mdl-31712323
14.
Evaluation of Dosimetry, Quantitative Methods, and Test-Retest Variability of 18F-PI-2620 PET for the Assessment of Tau Deposits in the Human Brain.
J Nucl Med
; 61(6): 920-927, 2020 06.
Artículo
en Inglés
| MEDLINE | ID: mdl-31712324
15.
Systematic comparison of two novel, thiol-reactive prosthetic groups for 18F labeling of peptides and proteins with the acylation agent succinimidyl-4-[18F]fluorobenzoate ([18F]SFB).
Amino Acids
; 36(2): 283-95, 2009 Feb.
Artículo
en Inglés
| MEDLINE | ID: mdl-18414978
16.
Direct labelling of peptides with 2-[18F]fluoro-2-deoxy-d-glucose ([18F]FDG).
Bioorg Med Chem Lett
; 19(18): 5426-8, 2009 Sep 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-19665892
17.
Radiation dosimetry of [18F]GP1 for imaging activated glycoprotein IIb/IIIa receptors with positron emission tomography in patients with acute thromboembolism.
Nucl Med Biol
; 72-73: 45-48, 2019.
Artículo
en Inglés
| MEDLINE | ID: mdl-31330411
18.
The Characterization of 18F-hGTS13 for Molecular Imaging of xC- Transporter Activity with PET.
J Nucl Med
; 60(12): 1812-1817, 2019 12.
Artículo
en Inglés
| MEDLINE | ID: mdl-31171595
19.
Assessment of Tumor Redox Status through (S)-4-(3-[18F]fluoropropyl)-L-Glutamic Acid PET Imaging of System xc - Activity.
Cancer Res
; 79(4): 853-863, 2019 02 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-30401715
20.
A phase 1, first-in-human study of 18F-GP1 positron emission tomography for imaging acute arterial thrombosis.
EJNMMI Res
; 9(1): 3, 2019 Jan 07.
Artículo
en Inglés
| MEDLINE | ID: mdl-30617563