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1.
Mitochondrial quality control proteases and their modulation for cancer therapy.
Med Res Rev
; 43(2): 399-436, 2023 03.
Artículo
en Inglés
| MEDLINE | ID: mdl-36208112
2.
Epigenetic changes in Mycobacterium tuberculosis and its host provide potential targets or biomarkers for drug discovery and clinical diagnosis.
Pharmacol Res
; 179: 106195, 2022 05.
Artículo
en Inglés
| MEDLINE | ID: mdl-35364247
3.
Biophysical and biochemical properties of PHGDH revealed by studies on PHGDH inhibitors.
Cell Mol Life Sci
; 79(1): 27, 2021 Dec 31.
Artículo
en Inglés
| MEDLINE | ID: mdl-34971423
4.
Ribosome-targeting antibacterial agents: Advances, challenges, and opportunities.
Med Res Rev
; 41(4): 1855-1889, 2021 07.
Artículo
en Inglés
| MEDLINE | ID: mdl-33501747
5.
Discovery of novel indolin-2-one compounds as potent inhibitors of HsClpP for cancer treatment.
Bioorg Chem
; 110: 104820, 2021 05.
Artículo
en Inglés
| MEDLINE | ID: mdl-33773224
6.
Discovery of novel inhibitors of human phosphoglycerate dehydrogenase by activity-directed combinatorial chemical synthesis strategy.
Bioorg Chem
; 115: 105159, 2021 10.
Artículo
en Inglés
| MEDLINE | ID: mdl-34298241
7.
Structure-activity relationship study of DEL-22379: ERK dimerization inhibitors with increased safety.
Mol Divers
; 25(2): 1051-1075, 2021 May.
Artículo
en Inglés
| MEDLINE | ID: mdl-32377992
8.
Design and synthesis of novel spirooxindole-indenoquinoxaline derivatives as novel tryptophanyl-tRNA synthetase inhibitors.
Mol Divers
; 24(4): 1043-1063, 2020 Nov.
Artículo
en Inglés
| MEDLINE | ID: mdl-31834547
9.
A Novel Small Molecule, ZY354, Inhibits Dental Caries-Associated Oral Biofilms.
Antimicrob Agents Chemother
; 63(5)2019 05.
Artículo
en Inglés
| MEDLINE | ID: mdl-30858201
10.
Discovery of novel anti-tuberculosis agents with pyrrolo[1,2-a]quinoxaline-based scaffold.
Bioorg Med Chem Lett
; 28(11): 2084-2090, 2018 06 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-29748048
11.
Design, synthesis and biological evaluation of novel pyrrole derivatives as potential ClpP1P2 inhibitor against Mycobacterium tuberculosis.
Bioorg Chem
; 80: 422-432, 2018 10.
Artículo
en Inglés
| MEDLINE | ID: mdl-30005200
12.
Transcriptional Repressor PtvR Regulates Phenotypic Tolerance to Vancomycin in Streptococcus pneumoniae.
J Bacteriol
; 199(14)2017 07 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-28484041
13.
Efficacy of the novel oxazolidinone compound FYL-67 for preventing biofilm formation by Staphylococcus aureus.
J Antimicrob Chemother
; 69(11): 3011-9, 2014 Nov.
Artículo
en Inglés
| MEDLINE | ID: mdl-24997316
14.
Discovery of novel bis-oxazolidinone compounds as potential potent and selective antitubercular agents.
Bioorg Med Chem Lett
; 24(6): 1496-501, 2014 Mar 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-24582981
15.
Synthesis and evaluation of amide side-chain modified Agomelatine analogues as potential antidepressant-like agents.
Bioorg Med Chem Lett
; 24(7): 1672-6, 2014 Apr 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-24631187
16.
Application of covalent modality in proximity-induced drug pharmacology: Early development, current strategy, and feature directions.
Eur J Med Chem
; 271: 116394, 2024 May 05.
Artículo
en Inglés
| MEDLINE | ID: mdl-38643668
17.
In vitro and in vivo enhancement effect of glabridin on the antibacterial activity of colistin, against multidrug resistant Escherichia coli strains.
Phytomedicine
; 130: 155732, 2024 Jul 25.
Artículo
en Inglés
| MEDLINE | ID: mdl-38776738
18.
Repurposing TAK875 as a novel STAT3 inhibitor for treating inflammatory bowel disease.
Biochem Pharmacol
; 219: 115957, 2024 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-38049007
19.
Exploration of novel isoxazole-fused quinone derivatives as anti-colorectal cancer agents through inhibiting STAT3 and elevating ROS level.
Eur J Med Chem
; 272: 116448, 2024 Jun 05.
Artículo
en Inglés
| MEDLINE | ID: mdl-38704936
20.
Design, Synthesis, and Biological Evaluation of 5-(5-Iodo-2-isopropyl-4-methoxyphenoxy)pyrimidine-2,4-diamine (AF-353) Derivatives as Novel DHFR Inhibitors against Staphylococcus aureus.
J Med Chem
; 67(6): 4757-4781, 2024 Mar 28.
Artículo
en Inglés
| MEDLINE | ID: mdl-38466654