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Synthesis and Structure-Activity Relationship Analysis of 5-HT7 Receptor Antagonists: Piperazin-1-yl Substituted Unfused Heterobiaryls.
Strekowski, Lucjan; Saczewski, Jaroslaw; Raux, Elizabeth A; Fernando, Nilmi T; Klenc, Jeff; Paranjpe, Shirish; Raszkiewicz, Aldona; Blake, Ava L; Ehalt, Adam J; Barnes, Samuel; Baranowski, Timothy C; Sullivan, Shannon M; Satala, Grzegorz; Bojarski, Andrzej J.
Afiliación
  • Strekowski L; Department of Chemistry, Georgia State University, Atlanta, Georgia, GA 30302, USA. lucjan@gsu.edu.
  • Saczewski J; Department of Chemical Technology of Drugs, Medical University of Gdansk, Aleja Generala Józefa Hallera 107, Gdansk 80-416, Poland. js@gumed.edu.pl.
  • Raux EA; Department of Chemistry, Georgia State University, Atlanta, Georgia, GA 30302, USA. earaux@gmail.com.
  • Fernando NT; Department of Chemistry, Georgia State University, Atlanta, Georgia, GA 30302, USA. fernando.nilmi@gmail.com.
  • Klenc J; Department of Chemistry, Georgia State University, Atlanta, Georgia, GA 30302, USA. jklenc@merchantgould.com.
  • Paranjpe S; Department of Chemistry, Georgia State University, Atlanta, Georgia, GA 30302, USA. shirishp007@gmail.com.
  • Raszkiewicz A; Department of Chemistry, Georgia State University, Atlanta, Georgia, GA 30302, USA. aldona.paluchowska@urpl.gov.pl.
  • Blake AL; Department of Chemistry, Georgia State University, Atlanta, Georgia, GA 30302, USA. ablake@bakerlaw.com.
  • Ehalt AJ; Department of Chemistry, Georgia State University, Atlanta, Georgia, GA 30302, USA. adamehalt@gmail.com.
  • Barnes S; Department of Chemistry, Georgia State University, Atlanta, Georgia, GA 30302, USA. sambarnes2@gmail.com.
  • Baranowski TC; Department of Chemistry, Georgia State University, Atlanta, Georgia, GA 30302, USA. tcb@bellsouth.net.
  • Sullivan SM; Department of Chemistry, Georgia State University, Atlanta, Georgia, GA 30302, USA. ssullivan@yahoo.com.
  • Satala G; Department of Medicinal Chemistry, Institute of Pharmacology, Polish Academy of Sciences, Smetna 12, Kraków 31-343, Poland. satala@if-pan.krakow.pl.
  • Bojarski AJ; Department of Medicinal Chemistry, Institute of Pharmacology, Polish Academy of Sciences, Smetna 12, Kraków 31-343, Poland. bojarski@if-pan.krakow.pl.
Molecules ; 21(4): 433, 2016 Mar 31.
Article en En | MEDLINE | ID: mdl-27043518

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Piperazinas / Antagonistas de la Serotonina / Relación Estructura-Actividad / Receptores de Serotonina Límite: Humans Idioma: En Revista: Molecules Asunto de la revista: BIOLOGIA Año: 2016 Tipo del documento: Article País de afiliación: Estados Unidos

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Piperazinas / Antagonistas de la Serotonina / Relación Estructura-Actividad / Receptores de Serotonina Límite: Humans Idioma: En Revista: Molecules Asunto de la revista: BIOLOGIA Año: 2016 Tipo del documento: Article País de afiliación: Estados Unidos