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Inhibitors to Overcome Secondary Mutations in the Stem Cell Factor Receptor KIT.
Kaitsiotou, Helena; Keul, Marina; Hardick, Julia; Mühlenberg, Thomas; Ketzer, Julia; Ehrt, Christiane; Krüll, Jasmin; Medda, Federico; Koch, Oliver; Giordanetto, Fabrizio; Bauer, Sebastian; Rauh, Daniel.
Afiliación
  • Kaitsiotou H; Faculty of Chemistry and Chemical Biology, TU Dortmund University , Otto-Hahn-Straße 4a, D-44227 Dortmund, Germany.
  • Keul M; Faculty of Chemistry and Chemical Biology, TU Dortmund University , Otto-Hahn-Straße 4a, D-44227 Dortmund, Germany.
  • Hardick J; Faculty of Chemistry and Chemical Biology, TU Dortmund University , Otto-Hahn-Straße 4a, D-44227 Dortmund, Germany.
  • Mühlenberg T; Department of Medical Oncology, Sarcoma Centre West German Cancer Centre University Duisburg-Essen, Medical School , Hufelandstraße 55, D-45122 Essen, Germany.
  • Ketzer J; Germany and German Cancer Consortium (DKTK), Partner Site University Hospital Essen , D-45147 Essen, Germany.
  • Ehrt C; Department of Medical Oncology, Sarcoma Centre West German Cancer Centre University Duisburg-Essen, Medical School , Hufelandstraße 55, D-45122 Essen, Germany.
  • Krüll J; Germany and German Cancer Consortium (DKTK), Partner Site University Hospital Essen , D-45147 Essen, Germany.
  • Medda F; Faculty of Chemistry and Chemical Biology, TU Dortmund University , Otto-Hahn-Straße 4a, D-44227 Dortmund, Germany.
  • Koch O; Faculty of Chemistry and Chemical Biology, TU Dortmund University , Otto-Hahn-Straße 4a, D-44227 Dortmund, Germany.
  • Giordanetto F; Taros Chemicals GmbH & Co. KG , Emil-Figge-Straße 76a, D-44227 Dortmund, Germany.
  • Bauer S; Faculty of Chemistry and Chemical Biology, TU Dortmund University , Otto-Hahn-Straße 4a, D-44227 Dortmund, Germany.
  • Rauh D; Taros Chemicals GmbH & Co. KG , Emil-Figge-Straße 76a, D-44227 Dortmund, Germany.
J Med Chem ; 60(21): 8801-8815, 2017 11 09.
Article en En | MEDLINE | ID: mdl-28991465

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Proteínas Proto-Oncogénicas c-kit / Resistencia a Antineoplásicos / Inhibidores de Proteínas Quinasas / Mutación Límite: Humans Idioma: En Revista: J Med Chem Asunto de la revista: QUIMICA Año: 2017 Tipo del documento: Article País de afiliación: Alemania

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Proteínas Proto-Oncogénicas c-kit / Resistencia a Antineoplásicos / Inhibidores de Proteínas Quinasas / Mutación Límite: Humans Idioma: En Revista: J Med Chem Asunto de la revista: QUIMICA Año: 2017 Tipo del documento: Article País de afiliación: Alemania