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A Novel Prodrug of a γ-Glutamylcyclotransferase Inhibitor Suppresses Cancer Cell Proliferation in vitro and Inhibits Tumor Growth in a Xenograft Mouse Model of Prostate Cancer.
Ii, Hiromi; Yoshiya, Taku; Nakata, Susumu; Taniguchi, Keiko; Hidaka, Koushi; Tsuda, Shugo; Mochizuki, Masayoshi; Nishiuchi, Yuji; Tsuda, Yuko; Ito, Kosei; Kageyama, Susumu; Yoshiki, Tatsuhiro.
Afiliación
  • Ii H; Department of Clinical Oncology, Kyoto Pharmaceutical University, Misasagi-Nakauchicho 5, Yamashina-ku, Kyoto, 607-8414, Japan.
  • Yoshiya T; Peptide Institute Inc., 7-2-9 Saito-Asagi, Ibaraki-shi, Osaka, 567-0085, Japan.
  • Nakata S; Department of Clinical Oncology, Kyoto Pharmaceutical University, Misasagi-Nakauchicho 5, Yamashina-ku, Kyoto, 607-8414, Japan.
  • Taniguchi K; Department of Clinical Oncology, Kyoto Pharmaceutical University, Misasagi-Nakauchicho 5, Yamashina-ku, Kyoto, 607-8414, Japan.
  • Hidaka K; Faculty of Pharmaceutical Sciences, Cooperative Research Center of Life Sciences, Kobe Gakuin University, 1-1-3 Minatojima, Chuo-ku, Kobe, 650-8586, Japan.
  • Tsuda S; Peptide Institute Inc., 7-2-9 Saito-Asagi, Ibaraki-shi, Osaka, 567-0085, Japan.
  • Mochizuki M; Peptide Institute Inc., 7-2-9 Saito-Asagi, Ibaraki-shi, Osaka, 567-0085, Japan.
  • Nishiuchi Y; Peptide Institute Inc., 7-2-9 Saito-Asagi, Ibaraki-shi, Osaka, 567-0085, Japan.
  • Tsuda Y; Present address: GlyTech Inc., 134 Chudoji Minamimachi, KRP #1-109, Shimogyo-ku, Kyoto, 600-8813, Japan.
  • Ito K; Faculty of Pharmaceutical Sciences, Cooperative Research Center of Life Sciences, Kobe Gakuin University, 1-1-3 Minatojima, Chuo-ku, Kobe, 650-8586, Japan.
  • Kageyama S; Graduate School of Biomedical Sciences, Nagasaki University, 1-7-1 Sakamoto, Nagasaki, 852-8588, Japan.
  • Yoshiki T; Department of Urology, Shiga University of Medical Science, Seta Tsukinowa-cho, Otsu, Shiga, 520-2192, Japan.
ChemMedChem ; 13(2): 155-163, 2018 01 22.
Article en En | MEDLINE | ID: mdl-29316360

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Neoplasias de la Próstata / Profármacos / Proliferación Celular / Dipéptidos / Gamma-Glutamilciclotransferasa / Antineoplásicos Límite: Animals / Humans / Male Idioma: En Revista: ChemMedChem Asunto de la revista: FARMACOLOGIA / QUIMICA Año: 2018 Tipo del documento: Article País de afiliación: Japón

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Neoplasias de la Próstata / Profármacos / Proliferación Celular / Dipéptidos / Gamma-Glutamilciclotransferasa / Antineoplásicos Límite: Animals / Humans / Male Idioma: En Revista: ChemMedChem Asunto de la revista: FARMACOLOGIA / QUIMICA Año: 2018 Tipo del documento: Article País de afiliación: Japón