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N-aryl-piperidine-4-carboxamides as a novel class of potent inhibitors of MALT1 proteolytic activity.
Schlapbach, Achim; Revesz, Laszlo; Pissot Soldermann, Carole; Zoller, Thomas; Régnier, Catherine H; Bornancin, Frédéric; Radimerski, Thomas; Blank, Jutta; Schuffenhauer, Ansgar; Renatus, Martin; Erbel, Paulus; Melkko, Samu; Heng, Richard; Simic, Oliver; Endres, Ralf; Wartmann, Markus; Quancard, Jean.
Afiliación
  • Schlapbach A; Novartis Institutes for BioMedical Research, CH-4002 Basel, Switzerland. Electronic address: achim.schlapbach@novartis.com.
  • Revesz L; Novartis Institutes for BioMedical Research, CH-4002 Basel, Switzerland.
  • Pissot Soldermann C; Novartis Institutes for BioMedical Research, CH-4002 Basel, Switzerland.
  • Zoller T; Novartis Institutes for BioMedical Research, CH-4002 Basel, Switzerland.
  • Régnier CH; Novartis Institutes for BioMedical Research, CH-4002 Basel, Switzerland.
  • Bornancin F; Novartis Institutes for BioMedical Research, CH-4002 Basel, Switzerland.
  • Radimerski T; Novartis Institutes for BioMedical Research, CH-4002 Basel, Switzerland.
  • Blank J; Novartis Institutes for BioMedical Research, CH-4002 Basel, Switzerland.
  • Schuffenhauer A; Novartis Institutes for BioMedical Research, CH-4002 Basel, Switzerland.
  • Renatus M; Novartis Institutes for BioMedical Research, CH-4002 Basel, Switzerland.
  • Erbel P; Novartis Institutes for BioMedical Research, CH-4002 Basel, Switzerland.
  • Melkko S; Novartis Institutes for BioMedical Research, CH-4002 Basel, Switzerland.
  • Heng R; Novartis Institutes for BioMedical Research, CH-4002 Basel, Switzerland.
  • Simic O; Novartis Institutes for BioMedical Research, CH-4002 Basel, Switzerland.
  • Endres R; Novartis Institutes for BioMedical Research, CH-4002 Basel, Switzerland.
  • Wartmann M; Novartis Institutes for BioMedical Research, CH-4002 Basel, Switzerland.
  • Quancard J; Novartis Institutes for BioMedical Research, CH-4002 Basel, Switzerland.
Bioorg Med Chem Lett ; 28(12): 2153-2158, 2018 07 01.
Article en En | MEDLINE | ID: mdl-29759726

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Piperidinas / Proteína 1 de la Translocación del Linfoma del Tejido Linfático Asociado a Mucosas / Antineoplásicos Límite: Animals / Humans Idioma: En Revista: Bioorg Med Chem Lett Asunto de la revista: BIOQUIMICA / QUIMICA Año: 2018 Tipo del documento: Article

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Piperidinas / Proteína 1 de la Translocación del Linfoma del Tejido Linfático Asociado a Mucosas / Antineoplásicos Límite: Animals / Humans Idioma: En Revista: Bioorg Med Chem Lett Asunto de la revista: BIOQUIMICA / QUIMICA Año: 2018 Tipo del documento: Article