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Identification and SAR exploration of a novel series of Legumain inhibitors.
Eddie, Sharon L; Gregson, Aaron; Graham, Emma; Burton, Stephanie; Harrison, Timothy; Burden, Roberta; Scott, Christopher J; Mullan, Paul B; Williams, Rich.
Afiliación
  • Eddie SL; CCRCB Drug Discovery Group, Centre for Cancer Research and Cell Biology, Queen's University Belfast, 97 Lisburn Rd., Belfast BT9 7BL, United Kingdom.
  • Gregson A; CCRCB Drug Discovery Group, Centre for Cancer Research and Cell Biology, Queen's University Belfast, 97 Lisburn Rd., Belfast BT9 7BL, United Kingdom.
  • Graham E; CCRCB Drug Discovery Group, Centre for Cancer Research and Cell Biology, Queen's University Belfast, 97 Lisburn Rd., Belfast BT9 7BL, United Kingdom.
  • Burton S; Almac Discovery, Health Sciences Building, Queen's University Belfast, 97 Lisburn Rd., Belfast BT9 7AE, United Kingdom.
  • Harrison T; Almac Discovery, Health Sciences Building, Queen's University Belfast, 97 Lisburn Rd., Belfast BT9 7AE, United Kingdom.
  • Burden R; School of Pharmacy, Queen's University Belfast, 97 Lisburn Rd., Belfast BT9 7BL, United Kingdom.
  • Scott CJ; School of Pharmacy, Queen's University Belfast, 97 Lisburn Rd., Belfast BT9 7BL, United Kingdom.
  • Mullan PB; CCRCB Drug Discovery Group, Centre for Cancer Research and Cell Biology, Queen's University Belfast, 97 Lisburn Rd., Belfast BT9 7BL, United Kingdom.
  • Williams R; CCRCB Drug Discovery Group, Centre for Cancer Research and Cell Biology, Queen's University Belfast, 97 Lisburn Rd., Belfast BT9 7BL, United Kingdom. Electronic address: rich.williams@qub.ac.uk.
Bioorg Med Chem Lett ; 29(12): 1546-1548, 2019 06 15.
Article en En | MEDLINE | ID: mdl-31005445

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Cisteína Endopeptidasas / Inhibidores de Cisteína Proteinasa Tipo de estudio: Diagnostic_studies Límite: Animals / Humans Idioma: En Revista: Bioorg Med Chem Lett Asunto de la revista: BIOQUIMICA / QUIMICA Año: 2019 Tipo del documento: Article País de afiliación: Reino Unido

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Cisteína Endopeptidasas / Inhibidores de Cisteína Proteinasa Tipo de estudio: Diagnostic_studies Límite: Animals / Humans Idioma: En Revista: Bioorg Med Chem Lett Asunto de la revista: BIOQUIMICA / QUIMICA Año: 2019 Tipo del documento: Article País de afiliación: Reino Unido