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Design, synthesis, antimicrobial, and DNA gyrase inhibitory properties of fluoroquinolone-dichloroacetic acid hybrids.
Seliem, Israa A; Panda, Siva S; Girgis, Adel S; Nagy, Yosra I; George, Riham F; Fayad, Walid; Fawzy, Nehmedo G; Ibrahim, Tarek S; Al-Mahmoudy, Amany M M; Sakhuja, Rajeev; Abdel-Samii, Zakaria K M.
Afiliación
  • Seliem IA; Department of Chemistry and Physics, Augusta University, Augusta, GA, USA.
  • Panda SS; Department of Pharmaceutical Organic Chemistry, Faculty of Pharmacy, Zagazig University, Zagazig, Egypt.
  • Girgis AS; Department of Chemistry and Physics, Augusta University, Augusta, GA, USA.
  • Nagy YI; Department of Pesticide Chemistry, National Research Centre, Giza, Egypt.
  • George RF; Microbiology and Immunology Department, Faculty of Pharmacy, Cairo University, Cairo, Egypt.
  • Fayad W; Pharmaceutical Chemistry Department, Faculty of Pharmacy, Cairo University, Cairo, Egypt.
  • Fawzy NG; Drug Bioassay-Cell Culture Laboratory, Pharmacognosy Department, National Research Centre, Giza, Egypt.
  • Ibrahim TS; Department of Pesticide Chemistry, National Research Centre, Giza, Egypt.
  • Al-Mahmoudy AMM; Department of Pharmaceutical Organic Chemistry, Faculty of Pharmacy, Zagazig University, Zagazig, Egypt.
  • Sakhuja R; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, King Abdulaziz University, Jeddah, Saudi Arabia.
  • Abdel-Samii ZKM; Department of Pharmaceutical Organic Chemistry, Faculty of Pharmacy, Zagazig University, Zagazig, Egypt.
Chem Biol Drug Des ; 95(2): 248-259, 2020 02.
Article en En | MEDLINE | ID: mdl-31623026

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Fluoroquinolonas / Ácido Dicloroacético / Inhibidores de Topoisomerasa II / Antibacterianos Idioma: En Revista: Chem Biol Drug Des Asunto de la revista: BIOQUIMICA / FARMACIA / FARMACOLOGIA Año: 2020 Tipo del documento: Article País de afiliación: Estados Unidos

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Fluoroquinolonas / Ácido Dicloroacético / Inhibidores de Topoisomerasa II / Antibacterianos Idioma: En Revista: Chem Biol Drug Des Asunto de la revista: BIOQUIMICA / FARMACIA / FARMACOLOGIA Año: 2020 Tipo del documento: Article País de afiliación: Estados Unidos