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C-2 phenyl replacements to obtain potent quinoline-based Staphylococcus aureus NorA inhibitors.
Felicetti, Tommaso; Mangiaterra, Gianmarco; Cannalire, Rolando; Cedraro, Nicholas; Pietrella, Donatella; Astolfi, Andrea; Massari, Serena; Tabarrini, Oriana; Manfroni, Giuseppe; Barreca, Maria Letizia; Cecchetti, Violetta; Biavasco, Francesca; Sabatini, Stefano.
Afiliación
  • Felicetti T; Department of Pharmaceutical Sciences, Chemistry and Technology of the Drug Section, Università degli Studi di Perugia, Perugia, Italy.
  • Mangiaterra G; Department of Life and Environmental Sciences, Università Politecnica delle Marche, Ancona, Italy.
  • Cannalire R; Department of Pharmaceutical Sciences, Chemistry and Technology of the Drug Section, Università degli Studi di Perugia, Perugia, Italy.
  • Cedraro N; Department of Life and Environmental Sciences, Università Politecnica delle Marche, Ancona, Italy.
  • Pietrella D; Department of Pharmaceutical Sciences, Biochemical Sciences and Health Section, Università degli Studi di Perugia, Perugia, Italy.
  • Astolfi A; Department of Pharmaceutical Sciences, Chemistry and Technology of the Drug Section, Università degli Studi di Perugia, Perugia, Italy.
  • Massari S; Department of Pharmaceutical Sciences, Chemistry and Technology of the Drug Section, Università degli Studi di Perugia, Perugia, Italy.
  • Tabarrini O; Department of Pharmaceutical Sciences, Chemistry and Technology of the Drug Section, Università degli Studi di Perugia, Perugia, Italy.
  • Manfroni G; Department of Pharmaceutical Sciences, Chemistry and Technology of the Drug Section, Università degli Studi di Perugia, Perugia, Italy.
  • Barreca ML; Department of Pharmaceutical Sciences, Chemistry and Technology of the Drug Section, Università degli Studi di Perugia, Perugia, Italy.
  • Cecchetti V; Department of Pharmaceutical Sciences, Chemistry and Technology of the Drug Section, Università degli Studi di Perugia, Perugia, Italy.
  • Biavasco F; Department of Life and Environmental Sciences, Università Politecnica delle Marche, Ancona, Italy.
  • Sabatini S; Department of Pharmaceutical Sciences, Chemistry and Technology of the Drug Section, Università degli Studi di Perugia, Perugia, Italy.
J Enzyme Inhib Med Chem ; 35(1): 584-597, 2020 Dec.
Article en En | MEDLINE | ID: mdl-31992093

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Quinolinas / Staphylococcus aureus / Proteínas Bacterianas / Proteínas Asociadas a Resistencia a Múltiples Medicamentos / Antibacterianos Idioma: En Revista: J Enzyme Inhib Med Chem Asunto de la revista: BIOQUIMICA / QUIMICA Año: 2020 Tipo del documento: Article País de afiliación: Italia

Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Quinolinas / Staphylococcus aureus / Proteínas Bacterianas / Proteínas Asociadas a Resistencia a Múltiples Medicamentos / Antibacterianos Idioma: En Revista: J Enzyme Inhib Med Chem Asunto de la revista: BIOQUIMICA / QUIMICA Año: 2020 Tipo del documento: Article País de afiliación: Italia