Development of an Acrylamide-Based Inhibitor of Protein <i>S</i>-Acylation.

Azizi, Saara-Anne; Lan, Tong; Delalande, Clémence; Kathayat, Rahul S; Banales Mejia, Fernando; Qin, Alice; Brookes, Noah; Sandoval, Perla Jasmine; Dickinson, Bryan C

Development of an Acrylamide-Based Inhibitor of Protein S-Acylation.

Azizi, Saara-Anne; Lan, Tong; Delalande, Clémence; Kathayat, Rahul S; Banales Mejia, Fernando; Qin, Alice; Brookes, Noah; Sandoval, Perla Jasmine; Dickinson, Bryan C.

Afiliación

Azizi SA; Department of Chemistry, The University of Chicago, Chicago, Illinois 60637, United States.
Lan T; Medical Scientist Training Program, Pritzker School of Medicine, The University of Chicago, Chicago, Illinois 60637, United States.
Delalande C; Department of Chemistry, The University of Chicago, Chicago, Illinois 60637, United States.
Kathayat RS; Department of Chemistry, The University of Chicago, Chicago, Illinois 60637, United States.
Banales Mejia F; Department of Chemistry, The University of Chicago, Chicago, Illinois 60637, United States.
Qin A; Department of Chemistry, The University of Chicago, Chicago, Illinois 60637, United States.
Brookes N; Department of Chemistry, The University of Chicago, Chicago, Illinois 60637, United States.
Sandoval PJ; Department of Chemistry, The University of Chicago, Chicago, Illinois 60637, United States.
Dickinson BC; Department of Chemistry, The University of Chicago, Chicago, Illinois 60637, United States.

ACS Chem Biol ; 16(8): 1546-1556, 2021 08 20.

Article en En | MEDLINE | ID: mdl-34309372

Asunto(s)

Acrilamidas/farmacología; Aciltransferasas/antagonistas & inhibidores; Antígenos CD36/metabolismo; Inhibidores Enzimáticos/farmacología; Acrilamidas/síntesis química; Acrilamidas/toxicidad; Acilación/efectos de los fármacos; Animales; Línea Celular Tumoral; Inhibidores Enzimáticos/síntesis química; Inhibidores Enzimáticos/toxicidad; Receptores ErbB/metabolismo; Humanos; Lipoilación/efectos de los fármacos; Ratones; Procesamiento Proteico-Postraduccional/efectos de los fármacos

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Texto completo: 1 Colección: 01-internacional Banco de datos: MEDLINE Asunto principal: Acrilamidas / Aciltransferasas / Antígenos CD36 / Inhibidores Enzimáticos Límite: Animals / Humans Idioma: En Revista: ACS Chem Biol Año: 2021 Tipo del documento: Article País de afiliación: Estados Unidos

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