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Bioorg Med Chem Lett
; 21(8): 2224-8, 2011 Apr 15.
Artigo
em Inglês
| MEDLINE
| ID: mdl-21441024
RESUMO
A new series of IGF-1R inhibitors related to hydantoins were identified from a lead originating from HTS. Their noncompetitive property as well as their slow binding characteristics provided a series of compounds with unique selectivity and excellent cellular activities.