1.
Bioorg Med Chem Lett
; 21(1): 92-6, 2011 Jan 01.
Artigo
em Inglês
| MEDLINE
| ID: mdl-21146408
RESUMO
The SAR around a V1b antagonist HTS hit 3 was explored to produce a series of thiazole sulfonamides as a lead series with selectivity over the related V1 and oxytocin receptors.