1.
Bioorg Med Chem Lett
; 14(13): 3477-80, 2004 Jul 05.
Artigo
em Inglês
| MEDLINE
| ID: mdl-15177456
RESUMO
A novel series of PAI-1 inhibitors containing an oxadiazolidinedione moiety were identified by high through-put screening. Optimization of substituents by parallel synthesis and the iterative design toward understanding structure-activity relationship to improve potency are described.