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Artigo em Inglês | MEDLINE | ID: mdl-8097546

RESUMO

A radioreceptor assay (RRA) was developed to determine plasma levels of amisulpride. In in vitro binding conditions, the RRA technique was sensitive (11.6 nmol/l) and reliable, with a high degree of precision. The reproducibility of the method through statistical coefficients was < 7%. This method was applied to a pilot pharmacokinetic study in rabbits following single i.v. administration of amisulpride at 10 mg/kg. The results obtained were compared with those obtained by high performance liquid chromatography method (HPLC) in order to assess the validity of this new RRA technique.


Assuntos
Antipsicóticos/farmacocinética , Antagonistas dos Receptores de Dopamina D2 , Sulpirida/análogos & derivados , Amissulprida , Animais , Antipsicóticos/farmacologia , Cromatografia Líquida de Alta Pressão , Corpo Estriado/efeitos dos fármacos , Corpo Estriado/metabolismo , Técnicas In Vitro , Masculino , Coelhos , Ensaio Radioligante , Ratos , Ratos Wistar , Receptores de Dopamina D2/metabolismo , Espiperona/farmacocinética , Sulpirida/farmacocinética , Sulpirida/farmacologia
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