Regioselective halogenation of 2-substituted-1,2,3-triazoles via sp2 C-H activation.
Org Biomol Chem
; 11(45): 7830-3, 2013 Dec 07.
Article
em En
| MEDLINE
| ID: mdl-24129498
ABSTRACT
A highly regioselective halogenation of 2-substituted-1,2,3-triazoles was developed via sp(2) C-H activation. This method is compatible with halogen atoms, as well as electron-donating and electron-withdrawing groups. Meanwhile, the strategy is also efficient for the synthesis of a key intermediate of Suvorexant.
Texto completo:
1
Coleções:
01-internacional
Base de dados:
MEDLINE
Assunto principal:
Triazóis
/
Hidrocarbonetos Halogenados
Idioma:
En
Revista:
Org Biomol Chem
Assunto da revista:
BIOQUIMICA
/
QUIMICA
Ano de publicação:
2013
Tipo de documento:
Article
País de afiliação:
China