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Domains for activation and inactivation in G protein-coupled receptors--a mutational analysis of constitutive activity of the adenosine A2B receptor.
Peeters, Miriam C; Li, Qilan; Elands, Rachel; van Westen, Gerard J P; Lenselink, Eelke B; Müller, Christa E; IJzerman, Adriaan P.
Afiliação
  • Peeters MC; Division of Medicinal Chemistry, Leiden Academic Centre for Drug Research, Leiden University, P.O. Box 9502, 2300 RA Leiden, The Netherlands. Electronic address: m.c.peeters@lacdr.leidenuniv.nl.
  • Li Q; Division of Medicinal Chemistry, Leiden Academic Centre for Drug Research, Leiden University, P.O. Box 9502, 2300 RA Leiden, The Netherlands.
  • Elands R; Division of Medicinal Chemistry, Leiden Academic Centre for Drug Research, Leiden University, P.O. Box 9502, 2300 RA Leiden, The Netherlands.
  • van Westen GJ; Division of Medicinal Chemistry, Leiden Academic Centre for Drug Research, Leiden University, P.O. Box 9502, 2300 RA Leiden, The Netherlands.
  • Lenselink EB; Division of Medicinal Chemistry, Leiden Academic Centre for Drug Research, Leiden University, P.O. Box 9502, 2300 RA Leiden, The Netherlands.
  • Müller CE; Pharmaceutical Institute, Pharmaceutical Chemistry I, Pharmaceutical Sciences Bonn (PSB), University of Bonn, An der Immenburg 4, D-53121 Bonn, Germany.
  • IJzerman AP; Division of Medicinal Chemistry, Leiden Academic Centre for Drug Research, Leiden University, P.O. Box 9502, 2300 RA Leiden, The Netherlands.
Biochem Pharmacol ; 92(2): 348-57, 2014 Nov 15.
Article em En | MEDLINE | ID: mdl-25179146

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Análise Mutacional de DNA / Proteínas de Saccharomyces cerevisiae / Receptor A2B de Adenosina / Mutação Tipo de estudo: Clinical_trials Idioma: En Revista: Biochem Pharmacol Ano de publicação: 2014 Tipo de documento: Article País de publicação: Reino Unido

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Análise Mutacional de DNA / Proteínas de Saccharomyces cerevisiae / Receptor A2B de Adenosina / Mutação Tipo de estudo: Clinical_trials Idioma: En Revista: Biochem Pharmacol Ano de publicação: 2014 Tipo de documento: Article País de publicação: Reino Unido