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Biochemical and behavioral effects of PDE10A inhibitors: Relationship to target site occupancy.
Li, Yu-Wen; Seager, Matthew A; Wojcik, Trevor; Heman, Karen; Molski, Thaddeus F; Fernandes, Alda; Langdon, Shaun; Pendri, Annapurna; Gerritz, Samuel; Tian, Yuan; Hong, Yang; Gallagher, Lizbeth; Merritt, James R; Zhang, Chongwu; Westphal, Ryan; Zaczek, Robert; Macor, John E; Bronson, Joanne J; Lodge, Nicholas J.
Afiliação
  • Li YW; Neuroscience Biology, Bristol-Myers Squibb, 5 Research Parkway, Wallingford, CT 06492-7660, USA. Electronic address: yu-wen.li@bms.com.
  • Seager MA; Neuroscience Biology, Bristol-Myers Squibb, 5 Research Parkway, Wallingford, CT 06492-7660, USA.
  • Wojcik T; Neuroscience Biology, Bristol-Myers Squibb, 5 Research Parkway, Wallingford, CT 06492-7660, USA.
  • Heman K; Neuroscience Biology, Bristol-Myers Squibb, 5 Research Parkway, Wallingford, CT 06492-7660, USA.
  • Molski TF; Neuroscience Biology, Bristol-Myers Squibb, 5 Research Parkway, Wallingford, CT 06492-7660, USA.
  • Fernandes A; Neuroscience Biology, Bristol-Myers Squibb, 5 Research Parkway, Wallingford, CT 06492-7660, USA.
  • Langdon S; Neuroscience Biology, Bristol-Myers Squibb, 5 Research Parkway, Wallingford, CT 06492-7660, USA.
  • Pendri A; Neuroscience Chemistry, Bristol-Myers Squibb, 5 Research Parkway, Wallingford, CT 06492-7660, USA.
  • Gerritz S; Neuroscience Chemistry, Bristol-Myers Squibb, 5 Research Parkway, Wallingford, CT 06492-7660, USA.
  • Tian Y; Radiosynthesis, Bristol-Myers Squibb, 5 Research Parkway, Wallingford, CT 06492-7660, USA.
  • Hong Y; Radiosynthesis, Bristol-Myers Squibb, 5 Research Parkway, Wallingford, CT 06492-7660, USA.
  • Gallagher L; Lead Evaluation, Bristol-Myers Squibb, 5 Research Parkway, Wallingford, CT 06492-7660, USA.
  • Merritt JR; Pharmacopeia Inc, 3000 Eastpark Boulevard, Cranbury, NJ 08512, USA.
  • Zhang C; Pharmacopeia Inc, 3000 Eastpark Boulevard, Cranbury, NJ 08512, USA.
  • Westphal R; Neuroscience Biology, Bristol-Myers Squibb, 5 Research Parkway, Wallingford, CT 06492-7660, USA.
  • Zaczek R; Neuroscience Biology, Bristol-Myers Squibb, 5 Research Parkway, Wallingford, CT 06492-7660, USA.
  • Macor JE; Neuroscience Chemistry, Bristol-Myers Squibb, 5 Research Parkway, Wallingford, CT 06492-7660, USA.
  • Bronson JJ; Neuroscience Chemistry, Bristol-Myers Squibb, 5 Research Parkway, Wallingford, CT 06492-7660, USA.
  • Lodge NJ; Neuroscience Biology, Bristol-Myers Squibb, 5 Research Parkway, Wallingford, CT 06492-7660, USA.
Neuropharmacology ; 102: 121-35, 2016 Mar.
Article em En | MEDLINE | ID: mdl-26522433

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Inibidores de Fosfodiesterase / Antipsicóticos / Comportamento Animal / Encéfalo Tipo de estudo: Prognostic_studies Limite: Animals Idioma: En Revista: Neuropharmacology Ano de publicação: 2016 Tipo de documento: Article País de publicação: Reino Unido

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Inibidores de Fosfodiesterase / Antipsicóticos / Comportamento Animal / Encéfalo Tipo de estudo: Prognostic_studies Limite: Animals Idioma: En Revista: Neuropharmacology Ano de publicação: 2016 Tipo de documento: Article País de publicação: Reino Unido