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Discovery of phenoxyindazoles and phenylthioindazoles as RORγ inverse agonists.
Ouvry, Gilles; Bouix-Peter, Claire; Ciesielski, Fabrice; Chantalat, Laurent; Christin, Olivier; Comino, Catherine; Duvert, Denis; Feret, Christophe; Harris, Craig S; Lamy, Laurent; Luzy, Anne-Pascale; Musicki, Branislav; Orfila, Danielle; Pascau, Jonathan; Parnet, Véronique; Perrin, Agnès; Pierre, Romain; Polge, Gaëlle; Raffin, Catherine; Rival, Yves; Taquet, Nathalie; Thoreau, Etienne; Hennequin, Laurent F.
Afiliação
  • Ouvry G; Galderma R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France.
  • Bouix-Peter C; Galderma R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France.
  • Ciesielski F; NovAliX, Bld Sébastien Brant, Bioparc, 67405 Illkirch Cedex, France.
  • Chantalat L; Galderma R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France.
  • Christin O; Galderma R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France.
  • Comino C; Galderma R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France.
  • Duvert D; Galderma R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France.
  • Feret C; Galderma R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France.
  • Harris CS; Galderma R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France.
  • Lamy L; Galderma R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France.
  • Luzy AP; Galderma R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France.
  • Musicki B; Galderma R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France.
  • Orfila D; Galderma R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France.
  • Pascau J; Galderma R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France.
  • Parnet V; Galderma R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France.
  • Perrin A; Galderma R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France.
  • Pierre R; Galderma R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France.
  • Polge G; Galderma R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France.
  • Raffin C; Galderma R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France.
  • Rival Y; Galderma R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France.
  • Taquet N; Galderma R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France.
  • Thoreau E; Galderma R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France.
  • Hennequin LF; Galderma R&D, Les Templiers 2400 Route des Colles, 06410 Biot, France.
Bioorg Med Chem Lett ; 26(23): 5802-5808, 2016 12 01.
Article em En | MEDLINE | ID: mdl-27815118

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Membro 3 do Grupo F da Subfamília 1 de Receptores Nucleares / Indazóis Limite: Humans Idioma: En Revista: Bioorg Med Chem Lett Assunto da revista: BIOQUIMICA / QUIMICA Ano de publicação: 2016 Tipo de documento: Article País de afiliação: França País de publicação: Reino Unido

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Membro 3 do Grupo F da Subfamília 1 de Receptores Nucleares / Indazóis Limite: Humans Idioma: En Revista: Bioorg Med Chem Lett Assunto da revista: BIOQUIMICA / QUIMICA Ano de publicação: 2016 Tipo de documento: Article País de afiliação: França País de publicação: Reino Unido