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Synthesis, COX-1/2 inhibition activities and molecular docking study of isothiazolopyridine derivatives.
Swiatek, Piotr; Strzelecka, Malgorzata; Urniaz, Rafal; Gebczak, Katarzyna; Gebarowski, Tomasz; Gasiorowski, Kazimierz; Malinka, Wieslaw.
Afiliação
  • Swiatek P; Department of Chemistry of Drugs, Wroclaw Medical University, Borowska 211, 50-556 Wroclaw, Poland. Electronic address: piotr.swiatek@umed.wroc.pl.
  • Strzelecka M; Department of Chemistry of Drugs, Wroclaw Medical University, Borowska 211, 50-556 Wroclaw, Poland.
  • Urniaz R; Department of Medicine, Institute for Medical Research, University of Cambridge, Cambridge Biomedical Campus, Addenbrooke's Hospital, Hills Rd, CB2 0SP Cambridge, UK.
  • Gebczak K; Department of Basic Medical Science, Wroclaw Medical University, Borowska 211, 50-556 Wroclaw, Poland.
  • Gebarowski T; Department of Basic Medical Science, Wroclaw Medical University, Borowska 211, 50-556 Wroclaw, Poland.
  • Gasiorowski K; Department of Basic Medical Science, Wroclaw Medical University, Borowska 211, 50-556 Wroclaw, Poland.
  • Malinka W; Department of Chemistry of Drugs, Wroclaw Medical University, Borowska 211, 50-556 Wroclaw, Poland.
Bioorg Med Chem ; 25(1): 316-326, 2017 01 01.
Article em En | MEDLINE | ID: mdl-27842798

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Piridinas / Tiazóis / Inibidores de Ciclo-Oxigenase Limite: Animals Idioma: En Revista: Bioorg Med Chem Assunto da revista: BIOQUIMICA / QUIMICA Ano de publicação: 2017 Tipo de documento: Article País de publicação: Reino Unido

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Piridinas / Tiazóis / Inibidores de Ciclo-Oxigenase Limite: Animals Idioma: En Revista: Bioorg Med Chem Assunto da revista: BIOQUIMICA / QUIMICA Ano de publicação: 2017 Tipo de documento: Article País de publicação: Reino Unido