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Pyrimidine-Based Inhibitors of Dynamin I GTPase Activity: Competitive Inhibition at the Pleckstrin Homology Domain.
Odell, Luke R; Abdel-Hamid, Mohammed K; Hill, Timothy A; Chau, Ngoc; Young, Kelly A; Deane, Fiona M; Sakoff, Jennette A; Andersson, Sofia; Daniel, James A; Robinson, Phillip J; McCluskey, Adam.
Afiliação
  • Odell LR; Chemistry, School of Environmental and Life Sciences, The University of Newcastle , Callaghan, New South Wales 2308, Australia.
  • Abdel-Hamid MK; Chemistry, School of Environmental and Life Sciences, The University of Newcastle , Callaghan, New South Wales 2308, Australia.
  • Hill TA; Department of Medicinal Chemistry, Faculty of Pharmacy, Assiut University , Assiut 71526, Egypt.
  • Chau N; Chemistry, School of Environmental and Life Sciences, The University of Newcastle , Callaghan, New South Wales 2308, Australia.
  • Young KA; Children's Medical Research Institute, The University of Sydney , 214 Hawkesbury Road, Westmead New South Wales 2145, Australia.
  • Deane FM; Chemistry, School of Environmental and Life Sciences, The University of Newcastle , Callaghan, New South Wales 2308, Australia.
  • Sakoff JA; Chemistry, School of Environmental and Life Sciences, The University of Newcastle , Callaghan, New South Wales 2308, Australia.
  • Andersson S; Experimental Therapeutics Group, Department of Medical Oncology, Calvary Mater Newcastle Hospital , Edith Street, Waratah, 2298, New South Wales Australia.
  • Daniel JA; Department of Biology and Chemical Engineering, Mälardalens University , Box 325, S-631 05, Eskilstuna, Sweden.
  • Robinson PJ; Children's Medical Research Institute, The University of Sydney , 214 Hawkesbury Road, Westmead New South Wales 2145, Australia.
  • McCluskey A; Children's Medical Research Institute, The University of Sydney , 214 Hawkesbury Road, Westmead New South Wales 2145, Australia.
J Med Chem ; 60(1): 349-361, 2017 01 12.
Article em En | MEDLINE | ID: mdl-27997171

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Pirimidinas / Dinamina I / Inibidores Enzimáticos / Domínios de Homologia à Plecstrina Limite: Humans Idioma: En Revista: J Med Chem Assunto da revista: QUIMICA Ano de publicação: 2017 Tipo de documento: Article País de afiliação: Austrália País de publicação: Estados Unidos

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Pirimidinas / Dinamina I / Inibidores Enzimáticos / Domínios de Homologia à Plecstrina Limite: Humans Idioma: En Revista: J Med Chem Assunto da revista: QUIMICA Ano de publicação: 2017 Tipo de documento: Article País de afiliação: Austrália País de publicação: Estados Unidos