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Capzimin is a potent and specific inhibitor of proteasome isopeptidase Rpn11.
Li, Jing; Yakushi, Tanya; Parlati, Francesco; Mackinnon, Andrew L; Perez, Christian; Ma, Yuyong; Carter, Kyle P; Colayco, Sharon; Magnuson, Gavin; Brown, Brock; Nguyen, Kevin; Vasile, Stefan; Suyama, Eigo; Smith, Layton H; Sergienko, Eduard; Pinkerton, Anthony B; Chung, Thomas D Y; Palmer, Amy E; Pass, Ian; Hess, Sonja; Cohen, Seth M; Deshaies, Raymond J.
Afiliação
  • Li J; Division of Biology and Biological Engineering, California Institute of Technology, Pasadena, California, USA.
  • Yakushi T; Proteome Exploration Laboratory, Beckman Institute, California Institute of Technology, Pasadena, California, USA.
  • Parlati F; Division of Biology and Biological Engineering, California Institute of Technology, Pasadena, California, USA.
  • Mackinnon AL; Division of Biology and Biological Engineering, California Institute of Technology, Pasadena, California, USA.
  • Perez C; Department of Chemistry and Biochemistry, University of California San Diego, La Jolla, California, USA.
  • Ma Y; Department of Chemistry and Biochemistry, University of California San Diego, La Jolla, California, USA.
  • Carter KP; Department of Chemistry and Biochemistry, University of Colorado Boulder, Boulder, Colorado, USA.
  • Colayco S; Conrad Prebys Center for Chemical Genomics at Sanford Burnham Prebys Medical Discovery Institute, La Jolla, California, USA.
  • Magnuson G; Conrad Prebys Center for Chemical Genomics at Sanford Burnham Prebys Medical Discovery Institute, La Jolla, California, USA.
  • Brown B; Conrad Prebys Center for Chemical Genomics at Sanford Burnham Prebys Medical Discovery Institute, La Jolla, California, USA.
  • Nguyen K; Sanford-Burnham Center for Chemical Genomics at Sanford-Burnham Medical Research Institute Lake Nona, Orlando, Florida, USA.
  • Vasile S; Sanford-Burnham Center for Chemical Genomics at Sanford-Burnham Medical Research Institute Lake Nona, Orlando, Florida, USA.
  • Suyama E; Sanford-Burnham Center for Chemical Genomics at Sanford-Burnham Medical Research Institute Lake Nona, Orlando, Florida, USA.
  • Smith LH; Sanford-Burnham Center for Chemical Genomics at Sanford-Burnham Medical Research Institute Lake Nona, Orlando, Florida, USA.
  • Sergienko E; Conrad Prebys Center for Chemical Genomics at Sanford Burnham Prebys Medical Discovery Institute, La Jolla, California, USA.
  • Pinkerton AB; Conrad Prebys Center for Chemical Genomics at Sanford Burnham Prebys Medical Discovery Institute, La Jolla, California, USA.
  • Chung TDY; Conrad Prebys Center for Chemical Genomics at Sanford Burnham Prebys Medical Discovery Institute, La Jolla, California, USA.
  • Palmer AE; Department of Chemistry and Biochemistry, University of Colorado Boulder, Boulder, Colorado, USA.
  • Pass I; Conrad Prebys Center for Chemical Genomics at Sanford Burnham Prebys Medical Discovery Institute, La Jolla, California, USA.
  • Hess S; Proteome Exploration Laboratory, Beckman Institute, California Institute of Technology, Pasadena, California, USA.
  • Cohen SM; Department of Chemistry and Biochemistry, University of California San Diego, La Jolla, California, USA.
  • Deshaies RJ; Division of Biology and Biological Engineering, California Institute of Technology, Pasadena, California, USA.
Nat Chem Biol ; 13(5): 486-493, 2017 05.
Article em En | MEDLINE | ID: mdl-28244987

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Quinolinas / Transativadores / Inibidores de Proteassoma Tipo de estudo: Prognostic_studies Limite: Humans Idioma: En Revista: Nat Chem Biol Assunto da revista: BIOLOGIA / QUIMICA Ano de publicação: 2017 Tipo de documento: Article País de afiliação: Estados Unidos País de publicação: Estados Unidos

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Quinolinas / Transativadores / Inibidores de Proteassoma Tipo de estudo: Prognostic_studies Limite: Humans Idioma: En Revista: Nat Chem Biol Assunto da revista: BIOLOGIA / QUIMICA Ano de publicação: 2017 Tipo de documento: Article País de afiliação: Estados Unidos País de publicação: Estados Unidos