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Discovery, Development, and Cellular Delivery of Potent and Selective Bicyclic Peptide Inhibitors of Grb7 Cancer Target.
Watson, Gabrielle M; Kulkarni, Ketav; Sang, Jianrong; Ma, Xiuquan; Gunzburg, Menachem J; Perlmutter, Patrick; Wilce, Matthew C J; Wilce, Jacqueline A.
Afiliação
  • Watson GM; Biomedicine Discovery Institute, Department of Biochemistry and Molecular Biology, Monash University , Wellington Road, Clayton, VIC 3800, Australia.
  • Kulkarni K; Biomedicine Discovery Institute, Department of Biochemistry and Molecular Biology, Monash University , Wellington Road, Clayton, VIC 3800, Australia.
  • Sang J; Biomedicine Discovery Institute, Department of Biochemistry and Molecular Biology, Monash University , Wellington Road, Clayton, VIC 3800, Australia.
  • Ma X; Department of Physiology, School of Medicine, Jiangsu University , Zhenjiang, Jiangsu 212013, P.R. China.
  • Gunzburg MJ; Biomedicine Discovery Institute, Department of Biochemistry and Molecular Biology, Monash University , Wellington Road, Clayton, VIC 3800, Australia.
  • Perlmutter P; Biomedicine Discovery Institute, Department of Biochemistry and Molecular Biology, Monash University , Wellington Road, Clayton, VIC 3800, Australia.
  • Wilce MCJ; School of Chemistry, Monash University , Wellington Road, Clayton, VIC 3800, Australia.
  • Wilce JA; Biomedicine Discovery Institute, Department of Biochemistry and Molecular Biology, Monash University , Wellington Road, Clayton, VIC 3800, Australia.
J Med Chem ; 60(22): 9349-9359, 2017 11 22.
Article em En | MEDLINE | ID: mdl-29083893

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Peptídeos Cíclicos / Proteína Adaptadora GRB7 Limite: Humans Idioma: En Revista: J Med Chem Assunto da revista: QUIMICA Ano de publicação: 2017 Tipo de documento: Article País de afiliação: Austrália

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Peptídeos Cíclicos / Proteína Adaptadora GRB7 Limite: Humans Idioma: En Revista: J Med Chem Assunto da revista: QUIMICA Ano de publicação: 2017 Tipo de documento: Article País de afiliação: Austrália