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Synthesis and biological evaluation of indazole-4,7-dione derivatives as novel BRD4 inhibitors.
Yoo, Minjin; Yoo, Miyoun; Kim, Ji Eun; Lee, Heung Kyoung; Lee, Chong Ock; Park, Chi Hoon; Jung, Kwan-Young.
Afiliação
  • Yoo M; Department of Medicinal Chemistry and Pharmacology, University of Science & Technology, Daejeon, 34113, Republic of Korea.
  • Yoo M; Bio & Drug Discovery Division, Korea Research Institute of Chemical Technology, 141 Gajeong-ro, Yuseong-gu, Daejeon, 34114, Republic of Korea.
  • Kim JE; Bio & Drug Discovery Division, Korea Research Institute of Chemical Technology, 141 Gajeong-ro, Yuseong-gu, Daejeon, 34114, Republic of Korea.
  • Lee HK; Bio & Drug Discovery Division, Korea Research Institute of Chemical Technology, 141 Gajeong-ro, Yuseong-gu, Daejeon, 34114, Republic of Korea.
  • Lee CO; Bio & Drug Discovery Division, Korea Research Institute of Chemical Technology, 141 Gajeong-ro, Yuseong-gu, Daejeon, 34114, Republic of Korea.
  • Park CH; Department of Medicinal Chemistry and Pharmacology, University of Science & Technology, Daejeon, 34113, Republic of Korea. chpark@krict.re.kr.
  • Jung KY; Bio & Drug Discovery Division, Korea Research Institute of Chemical Technology, 141 Gajeong-ro, Yuseong-gu, Daejeon, 34114, Republic of Korea. chpark@krict.re.kr.
Arch Pharm Res ; 41(1): 46-56, 2018 Jan.
Article em En | MEDLINE | ID: mdl-29103140

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Fatores de Transcrição / Proteínas Nucleares / Indazóis / Antineoplásicos Tipo de estudo: Prognostic_studies Limite: Animals / Female / Humans Idioma: En Revista: Arch Pharm Res Ano de publicação: 2018 Tipo de documento: Article País de publicação:

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Fatores de Transcrição / Proteínas Nucleares / Indazóis / Antineoplásicos Tipo de estudo: Prognostic_studies Limite: Animals / Female / Humans Idioma: En Revista: Arch Pharm Res Ano de publicação: 2018 Tipo de documento: Article País de publicação: