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Quantitative, Wide-Spectrum Kinase Profiling in Live Cells for Assessing the Effect of Cellular ATP on Target Engagement.
Vasta, James D; Corona, Cesear R; Wilkinson, Jennifer; Zimprich, Chad A; Hartnett, James R; Ingold, Morgan R; Zimmerman, Kristopher; Machleidt, Thomas; Kirkland, Thomas A; Huwiler, Kristin G; Ohana, Rachel Friedman; Slater, Michael; Otto, Paul; Cong, Mei; Wells, Carrow I; Berger, Benedict-Tilman; Hanke, Thomas; Glas, Carina; Ding, Ke; Drewry, David H; Huber, Kilian V M; Willson, Timothy M; Knapp, Stefan; Müller, Susanne; Meisenheimer, Poncho L; Fan, Frank; Wood, Keith V; Robers, Matthew B.
Afiliação
  • Vasta JD; Promega Corporation, 2800 Woods Hollow Road, Fitchburg, WI 53711, USA.
  • Corona CR; Promega Biosciences Incorporated, 277 Granada Drive, San Luis Obispo, CA 93401, USA.
  • Wilkinson J; Promega Corporation, 2800 Woods Hollow Road, Fitchburg, WI 53711, USA.
  • Zimprich CA; Promega Corporation, 2800 Woods Hollow Road, Fitchburg, WI 53711, USA.
  • Hartnett JR; Promega Corporation, 2800 Woods Hollow Road, Fitchburg, WI 53711, USA.
  • Ingold MR; Promega Corporation, 2800 Woods Hollow Road, Fitchburg, WI 53711, USA.
  • Zimmerman K; Promega Corporation, 2800 Woods Hollow Road, Fitchburg, WI 53711, USA.
  • Machleidt T; Promega Corporation, 2800 Woods Hollow Road, Fitchburg, WI 53711, USA.
  • Kirkland TA; Promega Biosciences Incorporated, 277 Granada Drive, San Luis Obispo, CA 93401, USA.
  • Huwiler KG; Promega Corporation, 2800 Woods Hollow Road, Fitchburg, WI 53711, USA.
  • Ohana RF; Promega Corporation, 2800 Woods Hollow Road, Fitchburg, WI 53711, USA.
  • Slater M; Promega Corporation, 2800 Woods Hollow Road, Fitchburg, WI 53711, USA.
  • Otto P; Promega Corporation, 2800 Woods Hollow Road, Fitchburg, WI 53711, USA.
  • Cong M; Promega Corporation, 2800 Woods Hollow Road, Fitchburg, WI 53711, USA.
  • Wells CI; Structural Genomics Consortium, UNC Eshelman School of Pharmacy, University of North Carolina at Chapel Hill, Chapel Hill, NC, USA.
  • Berger BT; Structural Genomics Consortium, Institute for Pharmaceutical Chemistry, Johann Wolfgang Goethe-University, Max-von-Laue-Straße 9, 60438 Frankfurt am Main, Germany; Structural Genomics Consortium, Buchmann Institute for Molecular Life Sciences, Johann Wolfgang Goethe-University, Max-von-Laue-Straße 1
  • Hanke T; Structural Genomics Consortium, Institute for Pharmaceutical Chemistry, Johann Wolfgang Goethe-University, Max-von-Laue-Straße 9, 60438 Frankfurt am Main, Germany.
  • Glas C; Structural Genomics Consortium, Nuffield Department of Medicine, University of Oxford, Oxford, UK; Target Discovery Institute, Nuffield Department of Medicine, University of Oxford, Oxford, UK.
  • Ding K; State Key Laboratory of Respiratory Diseases, Guangzhou Institutes of Biomedicine and Health, Chinese Academy of Sciences, 190 Kaiyuan Avenue, Guangzhou 510530, China; School of Pharmacy, Jinan University, 601 Huangpu Avenue West, Guangzhou 510632, China.
  • Drewry DH; Structural Genomics Consortium, UNC Eshelman School of Pharmacy, University of North Carolina at Chapel Hill, Chapel Hill, NC, USA.
  • Huber KVM; Structural Genomics Consortium, Nuffield Department of Medicine, University of Oxford, Oxford, UK; Target Discovery Institute, Nuffield Department of Medicine, University of Oxford, Oxford, UK.
  • Willson TM; Structural Genomics Consortium, UNC Eshelman School of Pharmacy, University of North Carolina at Chapel Hill, Chapel Hill, NC, USA.
  • Knapp S; Structural Genomics Consortium, Institute for Pharmaceutical Chemistry, Johann Wolfgang Goethe-University, Max-von-Laue-Straße 9, 60438 Frankfurt am Main, Germany; Structural Genomics Consortium, Buchmann Institute for Molecular Life Sciences, Johann Wolfgang Goethe-University, Max-von-Laue-Straße 1
  • Müller S; Structural Genomics Consortium, Buchmann Institute for Molecular Life Sciences, Johann Wolfgang Goethe-University, Max-von-Laue-Straße 15, 60438 Frankfurt am Main, Germany.
  • Meisenheimer PL; Promega Biosciences Incorporated, 277 Granada Drive, San Luis Obispo, CA 93401, USA.
  • Fan F; Promega Corporation, 2800 Woods Hollow Road, Fitchburg, WI 53711, USA.
  • Wood KV; Promega Corporation, 2800 Woods Hollow Road, Fitchburg, WI 53711, USA.
  • Robers MB; Promega Corporation, 2800 Woods Hollow Road, Fitchburg, WI 53711, USA. Electronic address: matt.robers@promega.com.
Cell Chem Biol ; 25(2): 206-214.e11, 2018 02 15.
Article em En | MEDLINE | ID: mdl-29174542

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Fosfotransferases / Trifosfato de Adenosina / Inibidores de Proteínas Quinases Limite: Humans Idioma: En Revista: Cell Chem Biol Ano de publicação: 2018 Tipo de documento: Article País de afiliação: Estados Unidos País de publicação: Estados Unidos

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Fosfotransferases / Trifosfato de Adenosina / Inibidores de Proteínas Quinases Limite: Humans Idioma: En Revista: Cell Chem Biol Ano de publicação: 2018 Tipo de documento: Article País de afiliação: Estados Unidos País de publicação: Estados Unidos