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Design, Synthesis, and Pharmacological Evaluation of Novel ß2/3 Subunit-Selective γ-Aminobutyric Acid Type A (GABAA) Receptor Modulators.
Stadler, Marco; Monticelli, Serena; Seidel, Thomas; Luger, Denise; Salzer, Isabella; Boehm, Stefan; Holzer, Wolfgang; Schwarzer, Christoph; Urban, Ernst; Khom, Sophia; Langer, Thierry; Pace, Vittorio; Hering, Steffen.
Afiliação
  • Stadler M; Department of Pharmacology and Toxicology , University of Vienna , Althanstraße 14 , 1090 Vienna , Austria.
  • Monticelli S; Department of Pharmaceutical Chemistry , University of Vienna , Althanstraße 14 , 1090 Vienna , Austria.
  • Seidel T; Department of Pharmaceutical Chemistry , University of Vienna , Althanstraße 14 , 1090 Vienna , Austria.
  • Luger D; Department of Pharmacology and Toxicology , University of Vienna , Althanstraße 14 , 1090 Vienna , Austria.
  • Salzer I; Department of Neurophysiology and Neuropharmacology , Medical University Vienna , Schwarzspanierstraße 17 , 1090 Vienna , Austria.
  • Boehm S; Department of Neurophysiology and Neuropharmacology , Medical University Vienna , Schwarzspanierstraße 17 , 1090 Vienna , Austria.
  • Holzer W; Department of Pharmaceutical Chemistry , University of Vienna , Althanstraße 14 , 1090 Vienna , Austria.
  • Schwarzer C; Department of Pharmacology , Medical University Innsbruck , Peter-Mayr-Straße 1a , 6020 Innsbruck , Austria.
  • Urban E; Department of Pharmaceutical Chemistry , University of Vienna , Althanstraße 14 , 1090 Vienna , Austria.
  • Khom S; Department of Pharmacology and Toxicology , University of Vienna , Althanstraße 14 , 1090 Vienna , Austria.
  • Langer T; Department of Neuroscience , The Scripps Research Institute , 10550 N Torrey Pines Road , La Jolla , California 92037 , United States.
  • Pace V; Department of Pharmaceutical Chemistry , University of Vienna , Althanstraße 14 , 1090 Vienna , Austria.
  • Hering S; Department of Pharmaceutical Chemistry , University of Vienna , Althanstraße 14 , 1090 Vienna , Austria.
J Med Chem ; 62(1): 317-341, 2019 01 10.
Article em En | MEDLINE | ID: mdl-30289721

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Desenho de Fármacos / Receptores de GABA-A / Amidas / Anticonvulsivantes Limite: Animals Idioma: En Revista: J Med Chem Assunto da revista: QUIMICA Ano de publicação: 2019 Tipo de documento: Article País de afiliação: Áustria País de publicação: Estados Unidos

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Desenho de Fármacos / Receptores de GABA-A / Amidas / Anticonvulsivantes Limite: Animals Idioma: En Revista: J Med Chem Assunto da revista: QUIMICA Ano de publicação: 2019 Tipo de documento: Article País de afiliação: Áustria País de publicação: Estados Unidos