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2-Aminoimidazole-based antagonists of the 5-HT6 receptor - A new concept in aminergic GPCR ligand design.
Hogendorf, Adam S; Hogendorf, Agata; Kurczab, Rafal; Kalinowska-Tluscik, Justyna; Popik, Piotr; Nikiforuk, Agnieszka; Krawczyk, Martyna; Satala, Grzegorz; Lenda, Tomasz; Knutelska, Joanna; Bugno, Ryszard; Staron, Jakub; Pietrus, Wojciech; Matloka, Mikolaj; Dubiel, Krzysztof; Moszczynski-Petkowski, Rafal; Pieczykolan, Jerzy; Wieczorek, Maciej; Pilarski, Boguslaw; Zajdel, Pawel; Bojarski, Andrzej J.
Afiliação
  • Hogendorf AS; Institute of Pharmacology, Polish Academy of Sciences, 12 Smetna Street, 30-343, Kraków, Poland. Electronic address: ahogen@if-pan.krakow.pl.
  • Hogendorf A; Institute of Pharmacology, Polish Academy of Sciences, 12 Smetna Street, 30-343, Kraków, Poland.
  • Kurczab R; Institute of Pharmacology, Polish Academy of Sciences, 12 Smetna Street, 30-343, Kraków, Poland.
  • Kalinowska-Tluscik J; Faculty of Chemistry, Jagiellonian University, 2 Gronostajowa Street, 30-387, Kraków, Poland.
  • Popik P; Institute of Pharmacology, Polish Academy of Sciences, 12 Smetna Street, 30-343, Kraków, Poland.
  • Nikiforuk A; Institute of Pharmacology, Polish Academy of Sciences, 12 Smetna Street, 30-343, Kraków, Poland.
  • Krawczyk M; Institute of Pharmacology, Polish Academy of Sciences, 12 Smetna Street, 30-343, Kraków, Poland.
  • Satala G; Institute of Pharmacology, Polish Academy of Sciences, 12 Smetna Street, 30-343, Kraków, Poland.
  • Lenda T; Institute of Pharmacology, Polish Academy of Sciences, 12 Smetna Street, 30-343, Kraków, Poland.
  • Knutelska J; Faculty of Pharmacy, Jagiellonian University Medical College, 9 Medyczna Street, 30-688, Kraków, Poland.
  • Bugno R; Institute of Pharmacology, Polish Academy of Sciences, 12 Smetna Street, 30-343, Kraków, Poland.
  • Staron J; Institute of Pharmacology, Polish Academy of Sciences, 12 Smetna Street, 30-343, Kraków, Poland.
  • Pietrus W; Institute of Pharmacology, Polish Academy of Sciences, 12 Smetna Street, 30-343, Kraków, Poland; Faculty of Chemistry, Jagiellonian University, 2 Gronostajowa Street, 30-387, Kraków, Poland.
  • Matloka M; Research & Development Centre, Celon Pharma S.A, 41A Mokra Street, Kielpin, 05-092, Lomianki, Poland.
  • Dubiel K; Research & Development Centre, Celon Pharma S.A, 41A Mokra Street, Kielpin, 05-092, Lomianki, Poland.
  • Moszczynski-Petkowski R; Research & Development Centre, Celon Pharma S.A, 41A Mokra Street, Kielpin, 05-092, Lomianki, Poland.
  • Pieczykolan J; Research & Development Centre, Celon Pharma S.A, 41A Mokra Street, Kielpin, 05-092, Lomianki, Poland.
  • Wieczorek M; Research & Development Centre, Celon Pharma S.A, 41A Mokra Street, Kielpin, 05-092, Lomianki, Poland.
  • Pilarski B; CERKO, 96/98 Zwyciestwa Avenue, 81-525, Gdynia, Poland.
  • Zajdel P; Faculty of Pharmacy, Jagiellonian University Medical College, 9 Medyczna Street, 30-688, Kraków, Poland.
  • Bojarski AJ; Institute of Pharmacology, Polish Academy of Sciences, 12 Smetna Street, 30-343, Kraków, Poland.
Eur J Med Chem ; 179: 1-15, 2019 Oct 01.
Article em En | MEDLINE | ID: mdl-31229883

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Antagonistas da Serotonina / Desenho de Fármacos / Receptores de Serotonina / Disfunção Cognitiva / Imidazóis Limite: Animals / Humans / Male Idioma: En Revista: Eur J Med Chem Ano de publicação: 2019 Tipo de documento: Article País de publicação: França

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Antagonistas da Serotonina / Desenho de Fármacos / Receptores de Serotonina / Disfunção Cognitiva / Imidazóis Limite: Animals / Humans / Male Idioma: En Revista: Eur J Med Chem Ano de publicação: 2019 Tipo de documento: Article País de publicação: França