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Bioisosteric ferrocenyl aminoquinoline-benzimidazole hybrids: Antimicrobial evaluation and mechanistic insights.
Baartzes, N; Stringer, T; Seldon, R; Warner, D F; Taylor, D; Wittlin, S; Chibale, K; Smith, G S.
Afiliação
  • Baartzes N; Department of Chemistry, University of Cape Town, Rondebosch, 7701, Cape Town, South Africa.
  • Stringer T; Department of Chemistry, University of Cape Town, Rondebosch, 7701, Cape Town, South Africa.
  • Seldon R; Drug Discovery and Development Centre (H3D), Institute of Infectious Disease and Molecular Medicine, University of Cape Town, Rondebosch, 7701, Cape Town, South Africa.
  • Warner DF; SAMRC/NHLS/UCT Molecular Mycobacteriology Research Unit, DST/NRF Centre of Excellence for Biomedical TB Research, Department of Clinical Laboratory Sciences, University of Cape Town, Rondebosch, 7701, Cape Town, South Africa; Wellcome Centre for Infectious Diseases Research in Africa, University of
  • Taylor D; H3D, Division of Clinical Pharmacology, Department of Medicine, University of Cape Town, Observatory, 7925, Cape Town, South Africa.
  • Wittlin S; Swiss Tropical and Public Health Institute, Socinstrasse 57, 4002, Basel, Switzerland; University of Basel, 4003, Basel, Switzerland.
  • Chibale K; Department of Chemistry, University of Cape Town, Rondebosch, 7701, Cape Town, South Africa; South African Medical Research Council, Drug Discovery and Development Research Unit, Department of Chemistry and Institute of Infectious Disease and Molecular Medicine, University of Cape Town, Rondebosch,
  • Smith GS; Department of Chemistry, University of Cape Town, Rondebosch, 7701, Cape Town, South Africa. Electronic address: gregory.smith@uct.ac.za.
Eur J Med Chem ; 180: 121-133, 2019 Oct 15.
Article em En | MEDLINE | ID: mdl-31301563

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Plasmodium falciparum / Quinolinas / Benzimidazóis / Compostos Ferrosos / Malária / Antibacterianos / Antimaláricos Limite: Animals Idioma: En Revista: Eur J Med Chem Ano de publicação: 2019 Tipo de documento: Article País de afiliação: África do Sul País de publicação: França

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Plasmodium falciparum / Quinolinas / Benzimidazóis / Compostos Ferrosos / Malária / Antibacterianos / Antimaláricos Limite: Animals Idioma: En Revista: Eur J Med Chem Ano de publicação: 2019 Tipo de documento: Article País de afiliação: África do Sul País de publicação: França