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Halogenated and di-substituted benzenesulfonamides as selective inhibitors of carbonic anhydrase isoforms.
Zaksauskas, Audrius; Capkauskaite, Edita; Jezepcikas, Linas; Linkuviene, Vaida; Paketuryte, Vaida; Smirnov, Alexey; Leitans, Janis; Kazaks, Andris; Dvinskis, Elviss; Manakova, Elena; Grazulis, Saulius; Tars, Kaspars; Matulis, Daumantas.
Afiliação
  • Zaksauskas A; Department of Biothermodynamics and Drug Design, Institute of Biotechnology, Life Sciences Center, Vilnius University, Sauletekio al. 7, Vilnius, LT, 10257, Lithuania.
  • Capkauskaite E; Department of Biothermodynamics and Drug Design, Institute of Biotechnology, Life Sciences Center, Vilnius University, Sauletekio al. 7, Vilnius, LT, 10257, Lithuania.
  • Jezepcikas L; Department of Biothermodynamics and Drug Design, Institute of Biotechnology, Life Sciences Center, Vilnius University, Sauletekio al. 7, Vilnius, LT, 10257, Lithuania.
  • Linkuviene V; Department of Biothermodynamics and Drug Design, Institute of Biotechnology, Life Sciences Center, Vilnius University, Sauletekio al. 7, Vilnius, LT, 10257, Lithuania.
  • Paketuryte V; Department of Biothermodynamics and Drug Design, Institute of Biotechnology, Life Sciences Center, Vilnius University, Sauletekio al. 7, Vilnius, LT, 10257, Lithuania.
  • Smirnov A; Department of Biothermodynamics and Drug Design, Institute of Biotechnology, Life Sciences Center, Vilnius University, Sauletekio al. 7, Vilnius, LT, 10257, Lithuania.
  • Leitans J; Latvian Biomedical Research and Study Centre, Ratsupites 1 k-1, Riga, LV, 1067, Latvia.
  • Kazaks A; Latvian Biomedical Research and Study Centre, Ratsupites 1 k-1, Riga, LV, 1067, Latvia.
  • Dvinskis E; Latvian Biomedical Research and Study Centre, Ratsupites 1 k-1, Riga, LV, 1067, Latvia.
  • Manakova E; Department of Protein - DNA Interactions, Institute of Biotechnology, Life Sciences Center, Vilnius University, Sauletekio al. 7, Vilnius, LT, 10257, Lithuania.
  • Grazulis S; Department of Protein - DNA Interactions, Institute of Biotechnology, Life Sciences Center, Vilnius University, Sauletekio al. 7, Vilnius, LT, 10257, Lithuania.
  • Tars K; Latvian Biomedical Research and Study Centre, Ratsupites 1 k-1, Riga, LV, 1067, Latvia.
  • Matulis D; Department of Biothermodynamics and Drug Design, Institute of Biotechnology, Life Sciences Center, Vilnius University, Sauletekio al. 7, Vilnius, LT, 10257, Lithuania. Electronic address: daumantas.matulis@bti.vu.lt.
Eur J Med Chem ; 185: 111825, 2020 Jan 01.
Article em En | MEDLINE | ID: mdl-31740053

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Sulfonamidas / Inibidores da Anidrase Carbônica / Anidrases Carbônicas Tipo de estudo: Prognostic_studies Limite: Humans Idioma: En Revista: Eur J Med Chem Ano de publicação: 2020 Tipo de documento: Article País de afiliação: Lituânia País de publicação: França

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Sulfonamidas / Inibidores da Anidrase Carbônica / Anidrases Carbônicas Tipo de estudo: Prognostic_studies Limite: Humans Idioma: En Revista: Eur J Med Chem Ano de publicação: 2020 Tipo de documento: Article País de afiliação: Lituânia País de publicação: França