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The European Federation for Medicinal Chemistry (EFMC) Best Practice Initiative: Validating Chemical Probes.
Quancard, Jean; Cox, Brian; Finsinger, Dirk; Guéret, Stéphanie M; Hartung, Ingo V; Koolman, Hannes F; Messinger, Josef; Sbardella, Gianluca; Laufer, Stefan.
Afiliação
  • Quancard J; Global Discovery Chemistry, Novartis Institute For Biomedical Research, Novartis Pharma AG Novartis Campus CH, 4056, Basel., Switzerland.
  • Cox B; Professor of Pharmaceutical Chemistry School of Life Sciences, University of Sussex, Brighton, BN1 9RH, UK.
  • Finsinger D; Medicinal Chemistry, Global R&D Merck Healthcare KGaA, Frankfurter Straße 250, 64293, Darmstadt, Germany.
  • Guéret SM; Medicinal Chemistry, Research and Early Development Cardiovascular, Renal and Metabolism, BioPharmaceuticals R&D AstraZeneca, Gothenburg, Sweden.
  • Hartung IV; Medicinal Chemistry, Global R&D Merck Healthcare KGaA, Frankfurter Straße 250, 64293, Darmstadt, Germany.
  • Koolman HF; Medicinal chemistry, Boehringer Ingelheim Pharma GmbH & Co. KG, Birkendorfer Straße 65 D, 88397, Biberach an der Riss, Germany.
  • Messinger J; Global Medicine Design Orionpharma, Orionintie 1, FI-02101, Espoo, Finland.
  • Sbardella G; Department of Pharmacy Epigenetic Med Chem Lab, University of Salerno, Via Giovanni Paolo II 132, I-84084, Fisciano, SA, Italy.
  • Laufer S; Pharmaceutical&Medicinal Chemistry, Institute of Pharmacy&Biochemistry, Tübingen Center for Academic Drug Discovery, Auf der Morgenstelle 8 D, 72070 Tuebingen, Germany.
ChemMedChem ; 15(24): 2388-2390, 2020 12 15.
Article em En | MEDLINE | ID: mdl-32881363
ABSTRACT
As part of an initiative aimed to share best practices in Medicinal Chemistry, the European Federation for Medicinal Chemistry (EFMC) is preparing a series of webinars and slide sets focused on the early phase of drug discovery. This educational material is freely accessible through the EFMC. The main target audiences are students or early career scientists and we also believe it will be valuable for experienced practitioners. The first of the series is focused on the generation and validation of high-quality chemical probes, which are critical for drug discovery and more broadly to further our understanding of human biology and disease.
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Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Sociedades Científicas / Agências Internacionais / Química Farmacêutica / Descoberta de Drogas / Webcasts como Assunto / Indicadores e Reagentes Tipo de estudo: Guideline Limite: Humans País/Região como assunto: Europa Idioma: En Revista: ChemMedChem Assunto da revista: FARMACOLOGIA / QUIMICA Ano de publicação: 2020 Tipo de documento: Article País de afiliação: Suíça

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Sociedades Científicas / Agências Internacionais / Química Farmacêutica / Descoberta de Drogas / Webcasts como Assunto / Indicadores e Reagentes Tipo de estudo: Guideline Limite: Humans País/Região como assunto: Europa Idioma: En Revista: ChemMedChem Assunto da revista: FARMACOLOGIA / QUIMICA Ano de publicação: 2020 Tipo de documento: Article País de afiliação: Suíça
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