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Discovery of potent glycogen synthase kinase 3/cholinesterase inhibitors with neuroprotection as potential therapeutic agent for Alzheimer's disease.
Jiang, Xueyang; Wang, Yang; Liu, Chang; Xing, Caiyi; Wang, Yingming; Lyu, Weiping; Wang, Saisai; Li, Qihang; Chen, Tingkai; Chen, Yao; Feng, Feng; Liu, Wenyuan; Sun, Haopeng.
Afiliação
  • Jiang X; Department of Natural Medicinal Chemistry, China Pharmaceutical University, Nanjing 211198, China; School of Pharmacy, China Pharmaceutical University, Nanjing 211198, China.
  • Wang Y; Department of Pharmaceutical Analysis, Key Laboratory of Drug Quality Control and Pharmacovigilance, China Pharmaceutical University, Nanjing 211198, China; School of Pharmacy, China Pharmaceutical University, Nanjing 211198, China.
  • Liu C; Department of Pharmaceutical Analysis, Key Laboratory of Drug Quality Control and Pharmacovigilance, China Pharmaceutical University, Nanjing 211198, China.
  • Xing C; School of Pharmacy, China Pharmaceutical University, Nanjing 211198, China.
  • Wang Y; Department of Pharmaceutical Analysis, Key Laboratory of Drug Quality Control and Pharmacovigilance, China Pharmaceutical University, Nanjing 211198, China.
  • Lyu W; Department of Pharmaceutical Analysis, Key Laboratory of Drug Quality Control and Pharmacovigilance, China Pharmaceutical University, Nanjing 211198, China.
  • Wang S; College of Life Science and Technology, China Pharmaceutical University, Nanjing 211198, China.
  • Li Q; Department of Medicinal Chemistry, China Pharmaceutical University, Nanjing 211198, China.
  • Chen T; Department of Natural Medicinal Chemistry, China Pharmaceutical University, Nanjing 211198, China.
  • Chen Y; School of Pharmacy, Nanjing University of Chinese Medicine, Nanjing 210023, China.
  • Feng F; Department of Natural Medicinal Chemistry, China Pharmaceutical University, Nanjing 211198, China; Jiangsu Food and Pharmaceutical Science College, No.4 Meicheng Road, Huai'an 223003, China. Electronic address: fengfeng@cpu.edu.cn.
  • Liu W; Department of Pharmaceutical Analysis, Key Laboratory of Drug Quality Control and Pharmacovigilance, China Pharmaceutical University, Nanjing 211198, China. Electronic address: liuwenyuan8506@163.com.
  • Sun H; Department of Medicinal Chemistry, China Pharmaceutical University, Nanjing 211198, China. Electronic address: sunhaopeng@163.com.
Bioorg Med Chem ; 30: 115940, 2021 01 15.
Article em En | MEDLINE | ID: mdl-33340937

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Piridinas / Tiazóis / Inibidores da Colinesterase / Fármacos Neuroprotetores / Inibidores de Proteínas Quinases / Doença de Alzheimer Limite: Humans Idioma: En Revista: Bioorg Med Chem Assunto da revista: BIOQUIMICA / QUIMICA Ano de publicação: 2021 Tipo de documento: Article País de afiliação: China País de publicação: Reino Unido

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Piridinas / Tiazóis / Inibidores da Colinesterase / Fármacos Neuroprotetores / Inibidores de Proteínas Quinases / Doença de Alzheimer Limite: Humans Idioma: En Revista: Bioorg Med Chem Assunto da revista: BIOQUIMICA / QUIMICA Ano de publicação: 2021 Tipo de documento: Article País de afiliação: China País de publicação: Reino Unido