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Discovery of N-aryl sulphonamide-quinazoline derivatives as anti-gastric cancer agents in vitro and in vivo via activating the Hippo signalling pathway.
Niu, Jin-Bo; Hua, Chun-Quan; Liu, Yuan; Yu, Guang-Xi; Yang, Jia-Jia; Li, Yin-Ru; Zhang, Yan-Bing; Qi, Ying-Qiu; Song, Jian; Jin, Cheng-Yun; Zhang, Sai-Yang.
Afiliação
  • Niu JB; The Third Affiliated Hospital of Zhengzhou University, Zhengzhou, China.
  • Hua CQ; School of Pharmaceutical Sciences, Institute of Drug Discovery & Development, Key Laboratory of Advanced Drug Preparation Technologies (Ministry of Education), Zhengzhou University, Zhengzhou, China.
  • Liu Y; School of Pharmaceutical Sciences, Institute of Drug Discovery & Development, Key Laboratory of Advanced Drug Preparation Technologies (Ministry of Education), Zhengzhou University, Zhengzhou, China.
  • Yu GX; School of Basic Medical Sciences, Zhengzhou University, Zhengzhou, China.
  • Yang JJ; Department of Pharmacy, Zhengzhou People's Hospital, Zhengzhou, China.
  • Li YR; The Third Affiliated Hospital of Zhengzhou University, Zhengzhou, China.
  • Zhang YB; School of Basic Medical Sciences, Zhengzhou University, Zhengzhou, China.
  • Qi YQ; School of Basic Medical Sciences, Zhengzhou University, Zhengzhou, China.
  • Song J; School of Pharmaceutical Sciences, Institute of Drug Discovery & Development, Key Laboratory of Advanced Drug Preparation Technologies (Ministry of Education), Zhengzhou University, Zhengzhou, China.
  • Jin CY; The Third Affiliated Hospital of Zhengzhou University, Zhengzhou, China.
  • Zhang SY; School of Pharmaceutical Sciences, Institute of Drug Discovery & Development, Key Laboratory of Advanced Drug Preparation Technologies (Ministry of Education), Zhengzhou University, Zhengzhou, China.
J Enzyme Inhib Med Chem ; 36(1): 1715-1731, 2021 Dec.
Article em En | MEDLINE | ID: mdl-34425716

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Quinazolinas / Neoplasias Gástricas / Sulfonamidas / Proteínas Serina-Treonina Quinases / Antineoplásicos Tipo de estudo: Prognostic_studies Limite: Animals / Humans Idioma: En Revista: J Enzyme Inhib Med Chem Assunto da revista: BIOQUIMICA / QUIMICA Ano de publicação: 2021 Tipo de documento: Article País de afiliação: China País de publicação: Reino Unido

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Quinazolinas / Neoplasias Gástricas / Sulfonamidas / Proteínas Serina-Treonina Quinases / Antineoplásicos Tipo de estudo: Prognostic_studies Limite: Animals / Humans Idioma: En Revista: J Enzyme Inhib Med Chem Assunto da revista: BIOQUIMICA / QUIMICA Ano de publicação: 2021 Tipo de documento: Article País de afiliação: China País de publicação: Reino Unido