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Metabolism guided optimization of peptidomimetics as non-covalent proteasome inhibitors for cancer treatment.
Cao, Yu; Tu, Yutong; Fu, Liping; Yu, Qian; Gao, Lixin; Zhang, Mengmeng; Zeng, Linghui; Zhang, Chong; Shao, Jiaan; Zhu, Huajian; Zhou, Yubo; Li, Jia; Zhang, Jiankang.
Afiliação
  • Cao Y; School of Medicine, Zhejiang University City College, Hangzhou, 310015, China; College of Pharmaceutical Sciences, Zhejiang University, Hangzhou, 310058, China.
  • Tu Y; State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai, 201203, China; University of Chinese Academy of Sciences, Beijing, 100049, China.
  • Fu L; Department of Pharmacy, Shaoxing TCM Hospital Affiliated to Zhejiang Chinese Medical University, Shaoxing, 312000, China.
  • Yu Q; School of Medicine, Zhejiang University City College, Hangzhou, 310015, China; College of Pharmaceutical Sciences, Zhejiang University, Hangzhou, 310058, China.
  • Gao L; State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai, 201203, China; School of Pharmaceutical Science, Jiangnan University, Wuxi, 214122, China.
  • Zhang M; State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai, 201203, China.
  • Zeng L; School of Medicine, Zhejiang University City College, Hangzhou, 310015, China.
  • Zhang C; School of Medicine, Zhejiang University City College, Hangzhou, 310015, China.
  • Shao J; School of Medicine, Zhejiang University City College, Hangzhou, 310015, China.
  • Zhu H; School of Medicine, Zhejiang University City College, Hangzhou, 310015, China.
  • Zhou Y; State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai, 201203, China; University of Chinese Academy of Sciences, Beijing, 100049, China; Zhongshan Institute for Drug Discovery, Shanghai Institute of Metria Medica, Chinese Academy of Scienc
  • Li J; State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai, 201203, China; University of Chinese Academy of Sciences, Beijing, 100049, China; Zhongshan Institute for Drug Discovery, Shanghai Institute of Metria Medica, Chinese Academy of Scienc
  • Zhang J; School of Medicine, Zhejiang University City College, Hangzhou, 310015, China. Electronic address: zhang_jk@zucc.edu.cn.
Eur J Med Chem ; 233: 114211, 2022 Apr 05.
Article em En | MEDLINE | ID: mdl-35218994

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Peptidomiméticos / Neoplasias / Antineoplásicos Limite: Humans Idioma: En Revista: Eur J Med Chem Ano de publicação: 2022 Tipo de documento: Article País de afiliação: China País de publicação: França

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Peptidomiméticos / Neoplasias / Antineoplásicos Limite: Humans Idioma: En Revista: Eur J Med Chem Ano de publicação: 2022 Tipo de documento: Article País de afiliação: China País de publicação: França