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Investigating the Structure-Activity Relationship of 1,2,4-Triazine G-Protein-Coupled Receptor 84 (GPR84) Antagonists.
Mahindra, Amit; Jenkins, Laura; Marsango, Sara; Huggett, Mark; Huggett, Margaret; Robinson, Lindsay; Gillespie, Jonathan; Rajamanickam, Muralikrishnan; Morrison, Angus; McElroy, Stuart; Tikhonova, Irina G; Milligan, Graeme; Jamieson, Andrew G.
Afiliação
  • Mahindra A; School of Chemistry, University of Glasgow, Joseph Black Building, University Avenue, Glasgow G12 8QQ, U.K.
  • Jenkins L; Centre for Translational Pharmacology, Institute of Molecular, Cell and Systems Biology, University of Glasgow, Davidson Building, Glasgow G12 8QQ, U.K.
  • Marsango S; Centre for Translational Pharmacology, Institute of Molecular, Cell and Systems Biology, University of Glasgow, Davidson Building, Glasgow G12 8QQ, U.K.
  • Huggett M; BioAscent Discovery Ltd., Newhouse, Lanarkshire ML1 5UH, U.K.
  • Huggett M; European Screening Centre, University of Dundee, Newhouse, Lanarkshire ML1 5UH, U.K.
  • Robinson L; BioAscent Discovery Ltd., Newhouse, Lanarkshire ML1 5UH, U.K.
  • Gillespie J; European Screening Centre, University of Dundee, Newhouse, Lanarkshire ML1 5UH, U.K.
  • Rajamanickam M; BioAscent Discovery Ltd., Newhouse, Lanarkshire ML1 5UH, U.K.
  • Morrison A; European Screening Centre, University of Dundee, Newhouse, Lanarkshire ML1 5UH, U.K.
  • McElroy S; BioAscent Discovery Ltd., Newhouse, Lanarkshire ML1 5UH, U.K.
  • Tikhonova IG; European Screening Centre, University of Dundee, Newhouse, Lanarkshire ML1 5UH, U.K.
  • Milligan G; BioAscent Discovery Ltd., Newhouse, Lanarkshire ML1 5UH, U.K.
  • Jamieson AG; European Screening Centre, University of Dundee, Newhouse, Lanarkshire ML1 5UH, U.K.
J Med Chem ; 65(16): 11270-11290, 2022 08 25.
Article em En | MEDLINE | ID: mdl-35948061

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Triazinas / Receptores Acoplados a Proteínas G Idioma: En Revista: J Med Chem Assunto da revista: QUIMICA Ano de publicação: 2022 Tipo de documento: Article País de afiliação: Reino Unido

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Triazinas / Receptores Acoplados a Proteínas G Idioma: En Revista: J Med Chem Assunto da revista: QUIMICA Ano de publicação: 2022 Tipo de documento: Article País de afiliação: Reino Unido