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Synthesis, Biochemical, and Cellular Evaluation of HDAC6 Targeting Proteolysis Targeting Chimeras.
Darwish, Salma; Heimburg, Tino; Ridinger, Johannes; Herp, Daniel; Schmidt, Matthias; Romier, Christophe; Jung, Manfred; Oehme, Ina; Sippl, Wolfgang.
Afiliação
  • Darwish S; Department of Medicinal Chemistry, Institute of Pharmacy, Martin-Luther University of Halle-Wittenberg, Halle/Saale, Germany.
  • Heimburg T; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Alexandria University, Alexandria, Egypt.
  • Ridinger J; Department of Medicinal Chemistry, Institute of Pharmacy, Martin-Luther University of Halle-Wittenberg, Halle/Saale, Germany.
  • Herp D; Hopp Children's Cancer Center Heidelberg (KiTZ), Heidelberg, Germany.
  • Schmidt M; Clinical Cooperation Unit Pediatric Oncology, German Cancer Research Center (DKFZ) and German Cancer Consortium (DKTK), Heidelberg, Germany.
  • Romier C; Institute of Pharmaceutical Sciences, University of Freiburg, Freiburg, Germany.
  • Jung M; Department of Medicinal Chemistry, Institute of Pharmacy, Martin-Luther University of Halle-Wittenberg, Halle/Saale, Germany.
  • Oehme I; Département de Biologie Structurale Intégrative, Université de Strasbourg, CNRS, INSERM, Institut de Génétique et de Biologie Moléculaire et Cellulaire (IGBMC), Illkirch Cedex, France.
  • Sippl W; Institute of Pharmaceutical Sciences, University of Freiburg, Freiburg, Germany.
Methods Mol Biol ; 2589: 179-193, 2023.
Article em En | MEDLINE | ID: mdl-36255625

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Complexo de Endopeptidases do Proteassoma / Neoplasias Limite: Humans Idioma: En Revista: Methods Mol Biol Assunto da revista: BIOLOGIA MOLECULAR Ano de publicação: 2023 Tipo de documento: Article País de afiliação: Alemanha País de publicação: Estados Unidos

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Complexo de Endopeptidases do Proteassoma / Neoplasias Limite: Humans Idioma: En Revista: Methods Mol Biol Assunto da revista: BIOLOGIA MOLECULAR Ano de publicação: 2023 Tipo de documento: Article País de afiliação: Alemanha País de publicação: Estados Unidos