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A non-traditional crystal-based compound screening method targeting the ATP binding site of Plasmodium falciparum GRP78 for identification of novel nucleoside analogues.
Mrozek, Alexander; Antoshchenko, Tetyana; Chen, Yun; Zepeda-Velázquez, Carlos; Smil, David; Kumar, Nirbhay; Lu, Hua; Park, Hee-Won.
Afiliação
  • Mrozek A; Department of Biochemistry & Molecular Biology, Tulane University School of Medicine, New Orleans, LA, United States.
  • Antoshchenko T; Department of Biochemistry & Molecular Biology, Tulane University School of Medicine, New Orleans, LA, United States.
  • Chen Y; Department of Biochemistry & Molecular Biology, Tulane University School of Medicine, New Orleans, LA, United States.
  • Zepeda-Velázquez C; Drug Discovery Program, Ontario Institute for Cancer Research, Toronto, ON, Canada.
  • Smil D; Drug Discovery Program, Ontario Institute for Cancer Research, Toronto, ON, Canada.
  • Kumar N; Department of Global Health, George Washington University Milken Institute of Public Health, Washington, D.C., DC, United States.
  • Lu H; Department of Biochemistry & Molecular Biology, Tulane University School of Medicine, New Orleans, LA, United States.
  • Park HW; Department of Biochemistry & Molecular Biology, Tulane University School of Medicine, New Orleans, LA, United States.
Front Mol Biosci ; 9: 956095, 2022.
Article em En | MEDLINE | ID: mdl-36275624

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Tipo de estudo: Diagnostic_studies / Screening_studies Idioma: En Revista: Front Mol Biosci Ano de publicação: 2022 Tipo de documento: Article País de afiliação: Estados Unidos País de publicação: Suíça

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Tipo de estudo: Diagnostic_studies / Screening_studies Idioma: En Revista: Front Mol Biosci Ano de publicação: 2022 Tipo de documento: Article País de afiliação: Estados Unidos País de publicação: Suíça