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Discovery of Potent Small-Molecule Inhibitors of WDR5-MYC Interaction.
Ding, Jian; Li, Guo; Liu, Hejun; Liu, Lulu; Lin, Ying; Gao, Jingyan; Zhou, Guoqiang; Shen, Lingling; Zhao, Mengxi; Yu, Yanyan; Guo, Weihui; Hommel, Ulrich; Ottl, Johannes; Blank, Jutta; Aubin, Nicola; Wei, Yi; He, Hu; Sage, David R; Atadja, Peter W; Li, En; Jain, Rishi K; Tallarico, John A; Canham, Stephen M; Chiang, Ying-Ling; Wang, He.
Afiliação
  • Ding J; Novartis Institutes for BioMedical Research, Cambridge, Massachusetts02139, United States.
  • Li G; Novartis Institutes for BioMedical Research, Shanghai201203, China.
  • Liu H; Novartis Institutes for BioMedical Research, Shanghai201203, China.
  • Liu L; Novartis Institutes for BioMedical Research, San Diego, California92121, United States.
  • Lin Y; Novartis Institutes for BioMedical Research, Cambridge, Massachusetts02139, United States.
  • Gao J; Novartis Institutes for BioMedical Research, Shanghai201203, China.
  • Zhou G; Novartis Institutes for BioMedical Research, Shanghai201203, China.
  • Shen L; Novartis Institutes for BioMedical Research, Shanghai201203, China.
  • Zhao M; Novartis Institutes for BioMedical Research, Cambridge, Massachusetts02139, United States.
  • Yu Y; Novartis Institutes for BioMedical Research, Shanghai201203, China.
  • Guo W; Novartis Institutes for BioMedical Research, Shanghai201203, China.
  • Hommel U; Novartis Institutes for BioMedical Research, Shanghai201203, China.
  • Ottl J; Novartis Institutes for BioMedical Research, Shanghai201203, China.
  • Blank J; Novartis Institutes for BioMedical Research, BaselCH-4056, Switzerland.
  • Aubin N; Novartis Institutes for BioMedical Research, BaselCH-4056, Switzerland.
  • Wei Y; Novartis Institutes for BioMedical Research, BaselCH-4056, Switzerland.
  • He H; Novartis Institutes for BioMedical Research, BaselCH-4056, Switzerland.
  • Sage DR; Novartis Institutes for BioMedical Research, Shanghai201203, China.
  • Atadja PW; Novartis Institutes for BioMedical Research, Shanghai201203, China.
  • Li E; Novartis Institutes for BioMedical Research, Cambridge, Massachusetts02139, United States.
  • Jain RK; Novartis Institutes for BioMedical Research, Shanghai201203, China.
  • Tallarico JA; Novartis Institutes for BioMedical Research, Shanghai201203, China.
  • Canham SM; Novartis Institutes for BioMedical Research, Cambridge, Massachusetts02139, United States.
  • Chiang YL; Novartis Institutes for BioMedical Research, Cambridge, Massachusetts02139, United States.
  • Wang H; Novartis Institutes for BioMedical Research, Cambridge, Massachusetts02139, United States.
ACS Chem Biol ; 18(1): 34-40, 2023 01 20.
Article em En | MEDLINE | ID: mdl-36594833

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Peptídeos e Proteínas de Sinalização Intracelular / Neoplasias Limite: Humans Idioma: En Revista: ACS Chem Biol Ano de publicação: 2023 Tipo de documento: Article País de afiliação: Estados Unidos País de publicação: Estados Unidos

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Peptídeos e Proteínas de Sinalização Intracelular / Neoplasias Limite: Humans Idioma: En Revista: ACS Chem Biol Ano de publicação: 2023 Tipo de documento: Article País de afiliação: Estados Unidos País de publicação: Estados Unidos