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Rational repurposing, synthesis, in vitro and in silico studies of chromone-peptidyl hybrids as potential agents against Leishmania donovani.
Hassan, Ahmed H E; Bayoumi, Waleed A; El-Sayed, Selwan M; Phan, Trong-Nhat; Kim, Yeon Ju; Lee, Chae Hyeon; Cho, Soo Bin; Oh, Taegeun; Ham, Gyeongpyo; Mahmoud, Kazem; No, Joo Hwan; Lee, Yong Sup.
Afiliação
  • Hassan AHE; Department of Medicinal Chemistry, Faculty of Pharmacy, Mansoura University, Mansoura, Egypt.
  • Bayoumi WA; Medicinal Chemistry Laboratory, Department of Pharmacy, College of Pharmacy, Kyung Hee University, Seoul, Republic of Korea.
  • El-Sayed SM; Department of Pharmaceutical Organic Chemistry, Faculty of Pharmacy, Mansoura University, Mansoura, Egypt.
  • Phan TN; Department of Medicinal Chemistry, Faculty of Pharmacy, Mansoura University, Mansoura, Egypt.
  • Kim YJ; Host-Parasite Research Laboratory, Institut Pasteur Korea, Gyeonggi-do, Republic of Korea.
  • Lee CH; Department of Fundamental Pharmaceutical Sciences, Kyung Hee University, Seoul, Republic of Korea.
  • Cho SB; Department of Fundamental Pharmaceutical Sciences, Kyung Hee University, Seoul, Republic of Korea.
  • Oh T; Department of Fundamental Pharmaceutical Sciences, Kyung Hee University, Seoul, Republic of Korea.
  • Ham G; Department of Fundamental Pharmaceutical Sciences, Kyung Hee University, Seoul, Republic of Korea.
  • Mahmoud K; Department of Fundamental Pharmaceutical Sciences, Kyung Hee University, Seoul, Republic of Korea.
  • No JH; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Egyptian Russian University, Badr City, Cairo, Egypt.
  • Lee YS; Host-Parasite Research Laboratory, Institut Pasteur Korea, Gyeonggi-do, Republic of Korea.
J Enzyme Inhib Med Chem ; 38(1): 2229071, 2023 Dec.
Article em En | MEDLINE | ID: mdl-37381756

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Leishmania donovani / Leishmaniose Visceral Tipo de estudo: Prognostic_studies Limite: Humans Idioma: En Revista: J Enzyme Inhib Med Chem Assunto da revista: BIOQUIMICA / QUIMICA Ano de publicação: 2023 Tipo de documento: Article País de afiliação: Egito País de publicação: Reino Unido

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Leishmania donovani / Leishmaniose Visceral Tipo de estudo: Prognostic_studies Limite: Humans Idioma: En Revista: J Enzyme Inhib Med Chem Assunto da revista: BIOQUIMICA / QUIMICA Ano de publicação: 2023 Tipo de documento: Article País de afiliação: Egito País de publicação: Reino Unido