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Macrocyclic Carbon-Linked Pyrazoles As Novel Inhibitors of MCL-1.
Demin, Samuël; Peschiulli, Aldo; Velter, Adriana I; Vos, Ann; De Boeck, Benoît; Miller, Bradley; Rombouts, Frederik J R; Reuillon, Tristan; Lento, William; Blanco, Maria Dominguez; Jouffroy, Matthieu; Steyvers, Helena; Bekkers, Mariette; Altrocchi, Cristina; Pietrak, Beth; Koo, Seong Joo; Szewczuk, Lawrence; Attar, Ricardo; Philippar, Ulrike.
Afiliação
  • Demin S; Janssen Research & Development, Janssen Pharmaceutica N.V., Turnhoutseweg 30, Beerse B-2340, Belgium.
  • Peschiulli A; Janssen Research & Development, Janssen Pharmaceutica N.V., Turnhoutseweg 30, Beerse B-2340, Belgium.
  • Velter AI; Janssen Research & Development, Janssen Pharmaceutica N.V., Turnhoutseweg 30, Beerse B-2340, Belgium.
  • Vos A; Janssen Research & Development, Janssen Pharmaceutica N.V., Turnhoutseweg 30, Beerse B-2340, Belgium.
  • De Boeck B; Janssen Research & Development, Janssen Pharmaceutica N.V., Turnhoutseweg 30, Beerse B-2340, Belgium.
  • Miller B; Janssen Research & Development LLC, 1400 McKean Road (Welsh Road), Spring House, Pennsylvania 19477, United States.
  • Rombouts FJR; Janssen Research & Development, Janssen Pharmaceutica N.V., Turnhoutseweg 30, Beerse B-2340, Belgium.
  • Reuillon T; Janssen Research & Development, Janssen Pharmaceutica N.V., Turnhoutseweg 30, Beerse B-2340, Belgium.
  • Lento W; Janssen Research & Development LLC, 1400 McKean Road (Welsh Road), Spring House, Pennsylvania 19477, United States.
  • Blanco MD; Janssen Research & Development, Janssen Pharmaceutica N.V., Turnhoutseweg 30, Beerse B-2340, Belgium.
  • Jouffroy M; Chemical Process R&D, Discovery Process Research, Janssen Pharmaceutica N.V., Beerse B-2340, Belgium.
  • Steyvers H; Janssen Research & Development, Janssen Pharmaceutica N.V., Turnhoutseweg 30, Beerse B-2340, Belgium.
  • Bekkers M; Janssen Research & Development, Janssen Pharmaceutica N.V., Turnhoutseweg 30, Beerse B-2340, Belgium.
  • Altrocchi C; Janssen Research & Development, Janssen Pharmaceutica N.V., Turnhoutseweg 30, Beerse B-2340, Belgium.
  • Pietrak B; Janssen Research & Development LLC, 1400 McKean Road (Welsh Road), Spring House, Pennsylvania 19477, United States.
  • Koo SJ; Janssen Research & Development, Janssen Pharmaceutica N.V., Turnhoutseweg 30, Beerse B-2340, Belgium.
  • Szewczuk L; Janssen Research & Development LLC, 1400 McKean Road (Welsh Road), Spring House, Pennsylvania 19477, United States.
  • Attar R; Janssen Research & Development LLC, 1400 McKean Road (Welsh Road), Spring House, Pennsylvania 19477, United States.
  • Philippar U; Janssen Research & Development, Janssen Pharmaceutica N.V., Turnhoutseweg 30, Beerse B-2340, Belgium.
ACS Med Chem Lett ; 14(7): 955-961, 2023 Jul 13.
Article em En | MEDLINE | ID: mdl-37465311

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Idioma: En Revista: ACS Med Chem Lett Ano de publicação: 2023 Tipo de documento: Article País de afiliação: Bélgica

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Idioma: En Revista: ACS Med Chem Lett Ano de publicação: 2023 Tipo de documento: Article País de afiliação: Bélgica