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Synthesis, Optimization, and Structure-Activity Relationships of Nicotinamide Phosphoribosyltransferase (NAMPT) Positive Allosteric Modulators (N-PAMs).
Shen, Zhengnan; Ratia, Kiira; Krider, Isabella; Ackerman-Berrier, Martha; Penton, Christopher; Musku, Soumya Reddy; Gordon-Blake, Jesse M; Laham, Megan S; Christie, Nicholas; Ma, Nina; Fu, Jiqiang; Xiong, Rui; Courey, Jenna M; Velma, Ganga Reddy; Thatcher, Gregory R J.
Afiliação
  • Shen Z; Department of Pharmacology and Toxicology, R. Ken Coit College of Pharmacy, University of Arizona, Tucson, Arizona 85721, United States.
  • Ratia K; Department of Pharmaceutical Sciences, College of Pharmacy, University of Illinois at Chicago, Chicago, Illinois 60612, United States.
  • Krider I; Research Resources Center, University of Illinois at Chicago, Chicago, Illinois 60612, United States.
  • Ackerman-Berrier M; Department of Chemistry & Biochemistry, Colleges of Science and Medicine, University of Arizona, Tucson, Arizona 85721, United States.
  • Penton C; Department of Pharmacology and Toxicology, R. Ken Coit College of Pharmacy, University of Arizona, Tucson, Arizona 85721, United States.
  • Musku SR; Department of Pharmacology and Toxicology, R. Ken Coit College of Pharmacy, University of Arizona, Tucson, Arizona 85721, United States.
  • Gordon-Blake JM; Department of Pharmacology and Toxicology, R. Ken Coit College of Pharmacy, University of Arizona, Tucson, Arizona 85721, United States.
  • Laham MS; Department of Pharmaceutical Sciences, College of Pharmacy, University of Illinois at Chicago, Chicago, Illinois 60612, United States.
  • Christie N; Department of Chemistry & Biochemistry, Colleges of Science and Medicine, University of Arizona, Tucson, Arizona 85721, United States.
  • Ma N; Department of Chemistry & Biochemistry, Colleges of Science and Medicine, University of Arizona, Tucson, Arizona 85721, United States.
  • Fu J; Department of Pharmacology and Toxicology, R. Ken Coit College of Pharmacy, University of Arizona, Tucson, Arizona 85721, United States.
  • Xiong R; Department of Pharmacology and Toxicology, R. Ken Coit College of Pharmacy, University of Arizona, Tucson, Arizona 85721, United States.
  • Courey JM; Department of Pharmacology and Toxicology, R. Ken Coit College of Pharmacy, University of Arizona, Tucson, Arizona 85721, United States.
  • Velma GR; Department of Chemistry & Biochemistry, Colleges of Science and Medicine, University of Arizona, Tucson, Arizona 85721, United States.
  • Thatcher GRJ; Department of Pharmacology and Toxicology, R. Ken Coit College of Pharmacy, University of Arizona, Tucson, Arizona 85721, United States.
J Med Chem ; 66(24): 16704-16727, 2023 12 28.
Article em En | MEDLINE | ID: mdl-38096366

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Nicotinamida Fosforribosiltransferase / NAD Idioma: En Revista: J Med Chem Assunto da revista: QUIMICA Ano de publicação: 2023 Tipo de documento: Article País de afiliação: Estados Unidos País de publicação: Estados Unidos

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Nicotinamida Fosforribosiltransferase / NAD Idioma: En Revista: J Med Chem Assunto da revista: QUIMICA Ano de publicação: 2023 Tipo de documento: Article País de afiliação: Estados Unidos País de publicação: Estados Unidos