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Discovery of a first-in-class protein degrader for the c-ros oncogene 1 (ROS1).
Yang, Jiawen; Wu, Yifan; Zhu, Qiaoliang; Qu, Xiaojuan; Ou, Hongyue; Liu, Haixia; Wei, Yongqi; Ge, Di; Lu, Chunlai; Jiang, Biao; Song, Xiaoling.
Afiliação
  • Yang J; Department of Thoracic Surgery, Zhongshan Hospital, Fudan University, Shanghai 200032, China; Shanghai Institute for Advanced Immunochemical Studies, ShanghaiTech University, Shanghai 201210, China; Shanghai Clinical Research and Trial Center, Shanghai 201210, China.
  • Wu Y; Shanghai Institute for Advanced Immunochemical Studies, ShanghaiTech University, Shanghai 201210, China; School of Life Science and Technology, ShanghaiTech University, Shanghai 201210, China.
  • Zhu Q; Department of Thoracic Surgery, Zhongshan Hospital, Fudan University, Shanghai 200032, China.
  • Qu X; Shanghai Institute for Advanced Immunochemical Studies, ShanghaiTech University, Shanghai 201210, China; School of Life Science and Technology, ShanghaiTech University, Shanghai 201210, China.
  • Ou H; Shanghai Institute for Advanced Immunochemical Studies, ShanghaiTech University, Shanghai 201210, China; School of Life Science and Technology, ShanghaiTech University, Shanghai 201210, China.
  • Liu H; Shanghai Institute for Advanced Immunochemical Studies, ShanghaiTech University, Shanghai 201210, China; School of Physical Science and Technology, ShanghaiTech University, Shanghai 201210, China.
  • Wei Y; Department of Thoracic Surgery, Zhongshan Hospital, Fudan University, Shanghai 200032, China.
  • Ge D; Department of Thoracic Surgery, Zhongshan Hospital, Fudan University, Shanghai 200032, China.
  • Lu C; Department of Thoracic Surgery, Zhongshan Hospital, Fudan University, Shanghai 200032, China. Electronic address: lu.chunlai@zs-hospital.sh.cn.
  • Jiang B; Shanghai Institute for Advanced Immunochemical Studies, ShanghaiTech University, Shanghai 201210, China; CAS Key Laboratory of Synthetic Chemistry of Natural Substances, Shanghai Institute of Organic Chemistry, Chinese Academy of Sciences, Shanghai 200032, China. Electronic address: jiangbiao@shangh
  • Song X; Shanghai Institute for Advanced Immunochemical Studies, ShanghaiTech University, Shanghai 201210, China. Electronic address: songxl@shanghaitech.edu.cn.
Bioorg Chem ; 150: 107590, 2024 Sep.
Article em En | MEDLINE | ID: mdl-38955003

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Proteínas Tirosina Quinases / Proteínas Proto-Oncogênicas / Proliferação de Células / Descoberta de Drogas / Antineoplásicos Limite: Animals / Humans Idioma: En Revista: Bioorg Chem Ano de publicação: 2024 Tipo de documento: Article País de afiliação: China País de publicação: Estados Unidos

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Proteínas Tirosina Quinases / Proteínas Proto-Oncogênicas / Proliferação de Células / Descoberta de Drogas / Antineoplásicos Limite: Animals / Humans Idioma: En Revista: Bioorg Chem Ano de publicação: 2024 Tipo de documento: Article País de afiliação: China País de publicação: Estados Unidos