Detalhe da pesquisa
1.
Development of Tyrphostin Analogues to Study Inhibition of the Mycobacterium tuberculosis Pup Proteasome System*.
Chembiochem
; 22(21): 3082-3089, 2021 11 03.
Artigo
Inglês
| MEDLINE | ID: mdl-34387015
2.
Escape from planarity in fragment-based drug discovery: A physicochemical and 3D property analysis of synthetic 3D fragment libraries.
Drug Discov Today Technol
; 38: 77-90, 2020 Dec.
Artigo
Inglês
| MEDLINE | ID: mdl-34895643
3.
Microwave-assisted diastereoselective two-step three-component synthesis for rapid access to drug-like libraries of substituted 3-amino-ß-lactams.
Bioorg Med Chem
; 26(1): 41-49, 2018 01 01.
Artigo
Inglês
| MEDLINE | ID: mdl-29174508
4.
Diastereoselective one-pot synthesis of tetrafunctionalized 2-imidazolines.
J Org Chem
; 79(11): 5219-26, 2014 Jun 06.
Artigo
Inglês
| MEDLINE | ID: mdl-24820129
5.
New Dual Inhibitors of Bacterial Topoisomerases with Broad-Spectrum Antibacterial Activity and In Vivo Efficacy against Vancomycin-Intermediate Staphylococcus aureus.
J Med Chem
; 66(6): 3968-3994, 2023 03 23.
Artigo
Inglês
| MEDLINE | ID: mdl-36877255
6.
Discovery and Hit-to-Lead Optimization of Benzothiazole Scaffold-Based DNA Gyrase Inhibitors with Potent Activity against Acinetobacter baumannii and Pseudomonas aeruginosa.
J Med Chem
; 66(2): 1380-1425, 2023 01 26.
Artigo
Inglês
| MEDLINE | ID: mdl-36634346
7.
Mycobacterium tuberculosis Proteasome Accessory Factor A (PafA) Can Transfer Prokaryotic Ubiquitin-Like Protein (Pup) between Substrates.
mBio
; 8(1)2017 02 21.
Artigo
Inglês
| MEDLINE | ID: mdl-28223451
8.
Chemoselective addition of isocyanides to N-tert-butanesulfinimines.
Org Lett
; 16(19): 5116-9, 2014 Oct 03.
Artigo
Inglês
| MEDLINE | ID: mdl-25229182