1.
J Labelled Comp Radiopharm
; 56(9-10): 461-3, 2013.
Artigo
em Inglês
| MEDLINE
| ID: mdl-24285521
RESUMO
The antitrypanosomal agent K777â¢HCl was labeled with carbon-14 to support absorption, distribution, metabolism, and excretion studies of this potential new drug for the treatment of Chagas disease. The radiolabeled compound was prepared in eight steps from [(14) C(U)]-(l)-phenylalanine with a specific activity of 54.4 mCi/mmol and an overall radiochemical yield of 4.1%.