1.
Bioorg Med Chem Lett
; 17(16): 4415-8, 2007 Aug 15.
Artigo
em Inglês
| MEDLINE
| ID: mdl-17590335
RESUMO
Rational replacement of the alkyne linker of mGluR5 antagonist MPEP gave 7-arylquinolines. SAR optimization gave an orally active compound with high affinity for the MPEP binding site.